SCHEMBL4647983

SCHEMBL4647983

Nc1cc(Oc2ccc(NC(=O)Nc3cc(C4CCCC4)nn3-c3ccc(Cl)cc3)cc2)ccn1

nearest known ligand 0.66

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KCNJ6 P48051 15/20 0.66
KCNJ3 P48549 15/20 0.66
KCNJ5 P48544 12/20 0.66
BRAF P15056 4/20 0.52
CYP3A4 P08684 1/20 0.47
GAA P10253 1/20 0.47
CYP2C19 P33261 1/20 0.47
MAPK14 Q16539 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4648677 0.85 MAPK14 (0.57) KCNJ6KCNJ3KCNJ5BRAFMAPK14
SCHEMBL2240721 0.85 KCNJ6 (0.58) KCNJ6KCNJ3KCNJ5BRAFCYP3A4
SCHEMBL2240958 0.83 KCNJ6 (0.56) KCNJ6KCNJ3KCNJ5BRAFCYP3A4
SCHEMBL2243108 0.81 MAPK14 (0.59) KCNJ6KCNJ3KCNJ5BRAFMAPK14
SCHEMBL4303949 0.80 KCNJ6 (0.58) KCNJ6KCNJ3KCNJ5BRAFMAPK14
SCHEMBL2246436 0.80 MAPK14 (0.59) KCNJ6KCNJ3KCNJ5BRAFMAPK14
SCHEMBL2243948 0.79 KCNJ6 (0.55) KCNJ6KCNJ3KCNJ5BRAFMAPK14
SCHEMBL13859627 0.79 KCNJ6 (0.69) KCNJ6KCNJ3KCNJ5BRAF
SCHEMBL2245642 0.78 KCNJ6 (0.60) KCNJ6KCNJ3KCNJ5BRAFMAPK14
SCHEMBL14537939 0.76 MAPK13 (0.62) BRAFMAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1960394-A2 PYRAZOLYL UREA DERIVATIVES USEFUL IN THE TREATMENT OF CANCER Bayer HealthCare AG (DE) 2008-08-27 EP disclosed
WO-2007059202-A2 PYRAZOLYL UREA DERIVATIVES USEFUL IN THE TREATMENT OF CANCER BAYER HEALTHCARE AG (DE) 2007-05-24 WO disclosed