SCHEMBL4648035

SCHEMBL4648035

Cc1ccc(-n2nc(C(C)(C)C)cc2NC(=O)Nc2ccc(Oc3ccnc(N)c3)cc2)cc1

nearest known ligand 0.79

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MAPK13 O15264 3/20 0.79
BRAF P15056 7/20 0.77
MAPK14 Q16539 6/20 0.77
PTK2 Q05397 5/20 0.66
ABL1 P00519 1/20 0.63
AXL P30530 1/20 0.63
MAPK12 P53778 1/20 0.63
MAPK11 Q15759 1/20 0.63
CYP2D6 P10635 2/20 0.61
CYP2C9 P11712 2/20 0.61
CYP2C8 P10632 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4648911 0.94 MAPK13 (0.69) MAPK13BRAFMAPK14PTK2ABL1
SCHEMBL4648598 0.94 MAPK13 (0.69) MAPK13BRAFMAPK14PTK2ABL1
SCHEMBL4689912 0.93 MAPK13 (0.68) MAPK13BRAFMAPK14PTK2ABL1
SCHEMBL14538174 0.93 MAPK13 (0.76) MAPK13BRAFMAPK14PTK2ABL1
SCHEMBL4689397 0.93 MAPK14 (0.69) MAPK13BRAFMAPK14ABL1AXL
SCHEMBL4691629 0.92 MAPK14 (0.69) MAPK13BRAFMAPK14ABL1AXL
SCHEMBL4788187 0.92 MAPK13 (0.67) MAPK13BRAFMAPK14PTK2ABL1
SCHEMBL4785151 0.91 MAPK13 (0.65) MAPK13BRAFMAPK14PTK2ABL1
SCHEMBL2243085 0.90 BRAF (0.84) MAPK13BRAFMAPK14PTK2ABL1
SCHEMBL4647839 0.90 MAPK13 (0.65) MAPK13BRAFMAPK14PTK2ABL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1960394-A2 PYRAZOLYL UREA DERIVATIVES USEFUL IN THE TREATMENT OF CANCER Bayer HealthCare AG (DE) 2008-08-27 EP disclosed
WO-2007059202-A2 PYRAZOLYL UREA DERIVATIVES USEFUL IN THE TREATMENT OF CANCER BAYER HEALTHCARE AG (DE) 2007-05-24 WO disclosed