SCHEMBL4648293

SCHEMBL4648293

CC(C)(C)c1cc(NC(=O)Nc2ccc(Oc3ccnc(N)c3)cc2)n(-c2ccc(F)c(F)c2)n1

nearest known ligand 0.68

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 9/20 0.68
MAPK13 O15264 4/20 0.64
BRAF P15056 7/20 0.62
ABL1 P00519 3/20 0.62
AXL P30530 1/20 0.62
SRC P12931 3/20 0.59
RAF1 P04049 1/20 0.55
MAPK12 P53778 1/20 0.53
MAPK11 Q15759 1/20 0.53
DDR2 Q16832 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4689912 0.91 MAPK13 (0.68) MAPK14MAPK13BRAFABL1AXL
SCHEMBL4648035 0.90 MAPK13 (0.79) MAPK14MAPK13BRAFABL1AXL
SCHEMBL4648837 0.89 MAPK14 (0.82) MAPK14MAPK13BRAFABL1AXL
SCHEMBL4648911 0.89 MAPK13 (0.69) MAPK14MAPK13BRAFABL1AXL
SCHEMBL4648404 0.88 MAPK13 (0.64) MAPK14MAPK13BRAFABL1AXL
SCHEMBL4689397 0.88 MAPK14 (0.69) MAPK14MAPK13BRAFABL1AXL
SCHEMBL14538174 0.88 MAPK13 (0.76) MAPK14MAPK13BRAFABL1AXL
SCHEMBL2243868 0.88 MAPK14 (0.82) MAPK14MAPK13BRAFABL1AXL
SCHEMBL4691629 0.87 MAPK14 (0.69) MAPK14MAPK13BRAFABL1AXL
SCHEMBL4788187 0.87 MAPK13 (0.67) MAPK14MAPK13BRAFABL1AXL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1960394-A2 PYRAZOLYL UREA DERIVATIVES USEFUL IN THE TREATMENT OF CANCER Bayer HealthCare AG (DE) 2008-08-27 EP disclosed
WO-2007059202-A2 PYRAZOLYL UREA DERIVATIVES USEFUL IN THE TREATMENT OF CANCER BAYER HEALTHCARE AG (DE) 2007-05-24 WO disclosed