SCHEMBL4649151

SCHEMBL4649151

Cc1ccc2c(c1)ncn2CCC(C)(C)NC[C@H](O)c1cccc(NS(=O)(=O)c2ccccc2)c1

nearest known ligand 0.47

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.47
NR1I2 O75469 14/20 0.46
ADRB3 P13945 2/20 0.45
HPGD P15428 1/20 0.45
KMT2A Q03164 2/20 0.42
MEN1 O00255 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4647480 0.94 ADRB3 (0.45) ALDH1A1NR1I2ADRB3HPGDKMT2A
SCHEMBL4605935 0.92 ADRB3 (0.46) ALDH1A1NR1I2ADRB3HPGDKMT2A
SCHEMBL1377347 0.91 NR1I2 (0.45) ALDH1A1NR1I2ADRB3HPGDKMT2A
SCHEMBL4914684 0.91 NR1I2 (0.44) ALDH1A1NR1I2ADRB3HPGDKMT2A
SCHEMBL1379764 0.91 NR1I2 (0.44) ALDH1A1NR1I2ADRB3HPGDKMT2A
SCHEMBL14185295 0.90 ADRB3 (0.48) ALDH1A1NR1I2ADRB3HPGDKMT2A
SCHEMBL14185294 0.89 ADRB3 (0.44) NR1I2ADRB3HPGDKMT2A
SCHEMBL1379766 0.89 ADRB3 (0.48) ALDH1A1NR1I2ADRB3HPGDKMT2A
SCHEMBL4908069 0.89 NR1I2 (0.43) ALDH1A1NR1I2ADRB3HPGDKMT2A
SCHEMBL4917492 0.89 NR1I2 (0.43) ALDH1A1NR1I2ADRB3HPGDKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1943229-A1 BENZIMIDAZOLE DERIVATIVES FOR USE AS BETA-3 RECEPTOR AGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-07-16 EP disclosed
WO-2007048842-A1 BENZIMIDAZOLE DERIVATIVES FOR USE AS BETA-3 RECEPTOR AGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2007-05-03 WO disclosed