SCHEMBL4647480

SCHEMBL4647480

Cc1ccc2ncn(CCC(C)(C)NC[C@H](O)c3cccc(NS(=O)(=O)c4ccccc4)c3)c2c1

nearest known ligand 0.45

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ADRB3 P13945 6/20 0.45
HPGD P15428 1/20 0.41
ALDH1A1 P00352 1/20 0.41
NR1I2 O75469 5/20 0.40
KMT2A Q03164 2/20 0.39
MEN1 O00255 1/20 0.39
HTR6 P50406 1/20 0.38
ADRB2 P07550 3/20 0.37
ADRB1 P08588 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4649151 0.94 ALDH1A1 (0.47) ADRB3HPGDALDH1A1NR1I2KMT2A
SCHEMBL4605935 0.92 ADRB3 (0.46) ADRB3HPGDALDH1A1NR1I2KMT2A
SCHEMBL4907424 0.91 ADRB3 (0.43) ADRB3HPGDNR1I2HTR6ADRB2
SCHEMBL4915375 0.91 ADRB3 (0.43) ADRB3HPGDNR1I2HTR6ADRB2
SCHEMBL4915362 0.91 ADRB3 (0.43) ADRB3HPGDNR1I2HTR6ADRB2
SCHEMBL14185295 0.90 ADRB3 (0.48) ADRB3HPGDALDH1A1NR1I2KMT2A
SCHEMBL14185294 0.89 ADRB3 (0.44) ADRB3HPGDNR1I2KMT2AHTR6
SCHEMBL4606660 0.89 NR1I2 (0.46) ADRB3HPGDNR1I2KMT2AMEN1
SCHEMBL4913365 0.88 ADRB3 (0.43) ADRB3HPGDALDH1A1KMT2AMEN1
SCHEMBL5468010 0.88 ADRB3 (0.43) ADRB3HPGDALDH1A1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1943229-A1 BENZIMIDAZOLE DERIVATIVES FOR USE AS BETA-3 RECEPTOR AGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-07-16 EP disclosed
WO-2007048842-A1 BENZIMIDAZOLE DERIVATIVES FOR USE AS BETA-3 RECEPTOR AGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2007-05-03 WO disclosed