SCHEMBL4649153

SCHEMBL4649153

NCC1CCN(Cc2ncc[nH]2)CC1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 1/20 0.67
HTR4 Q13639 1/20 0.45
CXCR4 P61073 1/20 0.44
PARP1 P09874 1/20 0.43
AKT2 P31751 3/20 0.43
GSK3B P49841 1/20 0.43
HTR2B P41595 3/20 0.39
KAT2B Q92831 1/20 0.38
ALDH1A1 P00352 2/20 0.37
OPRM1 P35372 1/20 0.37
GRIN2B Q13224 3/20 0.37
GRIN1 Q05586 1/20 0.36
KDM4E B2RXH2 1/20 0.36
LMNA P02545 1/20 0.36
HTR1D P28221 1/20 0.36
HTR1B P28222 1/20 0.36
GRIN2A Q12879 1/20 0.36
POLB P06746 1/20 0.36
GAA P10253 1/20 0.36
MAPT P10636 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4882040 0.98 ALOX15 (0.65) ALOX15HTR4CXCR4PARP1AKT2
SCHEMBL13512171 0.84 ALOX15 (0.67) ALOX15HTR4PARP1HTR2BKAT2B
SCHEMBL2675650 0.84 ALOX15 (0.71) ALOX15HTR4PARP1AKT2GSK3B
SCHEMBL15177859 0.82 ALOX15 (0.63) ALOX15HTR4PARP1HTR2BKAT2B
SCHEMBL15329166 0.81 ALOX15 (1.00) ALOX15HTR4PARP1KAT2BALDH1A1
SCHEMBL14375217 0.81 ALOX15 (0.71) ALOX15HTR4PARP1KAT2BALDH1A1
SCHEMBL13512449 0.81 ALOX15 (0.61) ALOX15HTR4CXCR4PARP1HTR2B
SCHEMBL8574775 0.79 GRIN2B (0.62) ALOX15HTR2BALDH1A1GRIN2BGRIN1
SCHEMBL1953418 0.78 ALOX15 (0.85) ALOX15PARP1KAT2BALDH1A1KDM4E
SCHEMBL4515060 0.78 ALOX15 (0.85) ALOX15PARP1KAT2BALDH1A1OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1904479-A2 NOVEL 2,4-DIANILINOPYRIMIDINE DERIVATIVES, THE PREPARATION THEREOF, THEIR USE AS MEDICAMENTS, PHARMACEUTICAL COMPOSITIONS AND, IN PARTICULAR, AS IKK INHIBITORS Sanofi-Aventis (FR) 2008-04-02 EP disclosed
WO-2007006926-A2 NOVEL 2,4-DIANILINOPYRIMIDINE DERIVATIVES, THE PREPARATION THEREOF, THEIR USE AS MEDICAMENTS, PHARMACEUTICAL COMPOSITIONS AND, IN PARTICULAR, AS IKK INHIBITORS SANOFI-AVENTIS (FR) 2007-01-18 WO disclosed