SCHEMBL4650643

SCHEMBL4650643

O=C(O)c1c[nH]c2c(F)c(Cc3cccc(OC(F)(F)F)c3)cc(F)c2c1=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM5A P29375 1/20 0.41
KDM4C Q9H3R0 1/20 0.41
KDM5B Q9UGL1 1/20 0.41
DAO P14920 1/20 0.39
FEN1 P39748 1/20 0.38
MPO P05164 1/20 0.38
RORC P51449 1/20 0.38
CYP2C9 P11712 1/20 0.37
MAPK14 Q16539 1/20 0.37
ROCK2 O75116 1/20 0.37
ROCK1 Q13464 1/20 0.37
DHODH Q02127 1/20 0.37
CSNK2A2 P19784 1/20 0.37
CSNK2B P67870 1/20 0.37
CSNK2A1 P68400 1/20 0.37
CDK2 P24941 1/20 0.36
MRGPRX4 Q96LA9 1/20 0.36
ALDH1A1 P00352 1/20 0.36
HPGD P15428 1/20 0.36
MDH2 P40926 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4650001 0.89 CSNK2A2 (0.39) DHODHCSNK2A2CSNK2BCSNK2A1CDK2
SCHEMBL4650011 0.88 KDM4C (0.45) KDM4CKDM5BCSNK2A2CSNK2BCSNK2A1
SCHEMBL4649980 0.86 CYP1A2 (0.43) DAODHODHCSNK2A2CSNK2BCSNK2A1
SCHEMBL4650110 0.81 KDM5A (0.42) KDM5AKDM4CKDM5BDAOCYP2C9
SCHEMBL4650790 0.81 KDM5A (0.42) KDM5AKDM5BDAOCSNK2A2CSNK2B
SCHEMBL4650109 0.81 CYP1A2 (0.46) KDM5AKDM4CKDM5BCSNK2A2CSNK2B
SCHEMBL4650035 0.80 CSNK2A2 (0.43) MAPK14CSNK2A2CSNK2BCSNK2A1ALDH1A1
SCHEMBL4650143 0.80 CSNK2A2 (0.43) CSNK2A2CSNK2BCSNK2A1ALDH1A1HPGD
SCHEMBL4559012 0.79 CHRM1 (0.43) CSNK2A2CSNK2BCSNK2A1ALDH1A1HPGD
SCHEMBL4649435 0.79 CLEC4M (0.47) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1963271-A1 QUINOLONE M1 RECEPTOR POSITIVE ALLOSTERIC MODULATORS Merck & Co., Inc. (US) 2008-09-03 EP claimed
WO-2007067489-A1 QUINOLONE M1 RECEPTOR POSITIVE ALLOSTERIC MODULATORS MERCK & CO., INC. (US) 2007-06-14 WO claimed