SCHEMBL4649980

SCHEMBL4649980

O=C(O)c1c[nH]c2c(F)c(Cc3cccc(C(F)(F)F)c3)cc(F)c2c1=O

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.43
MEN1 O00255 1/20 0.43
ALDH1A1 P00352 1/20 0.43
HPGD P15428 1/20 0.43
ALOX12 P18054 1/20 0.43
KMT2A Q03164 1/20 0.43
BACE1 P56817 1/20 0.40
NR4A2 P43354 2/20 0.39
DAO P14920 2/20 0.38
MRGPRX4 Q96LA9 2/20 0.38
CSNK2A2 P19784 1/20 0.38
CSNK2B P67870 1/20 0.38
CSNK2A1 P68400 1/20 0.38
HSD17B10 Q99714 1/20 0.38
RAB9A P51151 1/20 0.37
DHODH Q02127 1/20 0.37
PPARG P37231 1/20 0.37
PPARA Q07869 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4650109 0.89 CYP1A2 (0.46) CYP1A2MEN1ALDH1A1HPGDALOX12
SCHEMBL4650643 0.86 KDM5A (0.41) ALDH1A1HPGDDAOMRGPRX4CSNK2A2
SCHEMBL4650124 0.85 ALDH1A1 (0.47) CYP1A2MEN1ALDH1A1HPGDALOX12
SCHEMBL4650011 0.84 KDM4C (0.45) MEN1ALDH1A1HPGDKMT2ACSNK2A2
SCHEMBL4650790 0.83 KDM5A (0.42) CYP1A2ALDH1A1HPGDDAOCSNK2A2
SCHEMBL4650143 0.82 CSNK2A2 (0.43) CYP1A2ALDH1A1HPGDCSNK2A2CSNK2B
SCHEMBL4650035 0.82 CSNK2A2 (0.43) CYP1A2ALDH1A1HPGDCSNK2A2CSNK2B
SCHEMBL4650008 0.81 CSNK2A2 (0.39) CYP1A2MEN1ALDH1A1HPGDALOX12
SCHEMBL4559012 0.81 CHRM1 (0.43) CYP1A2ALDH1A1HPGDCSNK2A2CSNK2B
SCHEMBL4650012 0.80 PNP (0.41) CYP1A2HPGDCSNK2A2CSNK2BCSNK2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1963271-A1 QUINOLONE M1 RECEPTOR POSITIVE ALLOSTERIC MODULATORS Merck & Co., Inc. (US) 2008-09-03 EP claimed
WO-2007067489-A1 QUINOLONE M1 RECEPTOR POSITIVE ALLOSTERIC MODULATORS MERCK & CO., INC. (US) 2007-06-14 WO claimed