SCHEMBL4650939

SCHEMBL4650939

CC(OC(=O)Nc1ccccc1)C(=O)NC(CC(=O)O)C(O)CF

nearest known ligand 0.67

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 9/20 0.67
CASP7 P55210 1/20 0.53
CASP9 P55211 1/20 0.53
CASP6 P55212 1/20 0.53
CASP8 Q14790 1/20 0.53
KLK7 P49862 6/20 0.44
PSEN1 P49768 1/20 0.39
PSEN2 P49810 1/20 0.39
APH1B Q8WW43 1/20 0.39
NCSTN Q92542 1/20 0.39
APH1A Q96BI3 1/20 0.39
PSENEN Q9NZ42 1/20 0.39
ALDH1A1 P00352 1/20 0.37
LMNA P02545 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4650938 1.00 CASP3 (0.67) CASP3CASP7CASP9CASP6CASP8
SCHEMBL4650929 0.87 CASP3 (0.54) CASP3CASP7CASP9CASP6CASP8
SCHEMBL4650932 0.87 CASP3 (0.54) CASP3CASP7CASP9CASP6CASP8
SCHEMBL12569676 0.80 CASP3 (1.00) CASP3CASP7CASP9CASP6CASP8
SCHEMBL13914039 0.73 CASP3 (0.41) CASP3CASP7CASP9CASP6CASP8
SCHEMBL4426250 0.72 CASP3 (0.58) CASP3CASP7CASP9CASP6CASP8
SCHEMBL985454 0.72 CASP3 (0.56) CASP3CASP7CASP9CASP6CASP8
SCHEMBL54187 0.72 CASP3 (0.56) CASP3CASP7CASP9CASP6CASP8
SCHEMBL2811832 0.72 CASP3 (0.56) CASP3CASP7CASP9CASP6CASP8
SCHEMBL16899692 0.72 CASP3 (0.56) CASP3CASP7CASP9CASP6CASP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1212295-B1 SUBSTITUTED ALPHA-HYDROXY ACID CASPASE INHIBITORS AND THE USE THEREOF CYTOVIA INC (US) 2008-10-01 EP disclosed