SCHEMBL4654908

SCHEMBL4654908

CC(=O)Nc1cccc(-c2cc[c]cc2C(N)=O)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PI4K2A Q9BTU6 1/20 0.52
PARP1 P09874 1/20 0.47
DHODH Q02127 1/20 0.47
NQO2 P16083 2/20 0.46
CHEK2 O96017 1/20 0.46
ALDH1A1 P00352 2/20 0.46
BTK Q06187 1/20 0.45
BRD4 O60885 1/20 0.44
NPC1 O15118 3/20 0.43
RAB9A P51151 3/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
FYN P06241 2/20 0.43
TP53 P04637 1/20 0.43
STAT1 P42224 1/20 0.43
CYP1A2 P05177 1/20 0.43
HSD17B10 Q99714 1/20 0.43
TSHR P16473 1/20 0.43
KDM4E B2RXH2 1/20 0.43
GAA P10253 1/20 0.43
USP7 Q93009 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3225405 0.84 SMN1; SMN2 (0.50) PARP1DHODHALDH1A1BRD4RAB9A
SCHEMBL5605821 0.82 PI4K2A (0.57) PI4K2APARP1DHODHNQO2CHEK2
SCHEMBL27799605 0.81 NQO2 (0.45) PI4K2ANQO2ALDH1A1BRD4NPC1
SCHEMBL4631064 0.80 TLR8 (0.45) PARP1DHODHALDH1A1BRD4RAB9A
SCHEMBL16719394 0.78 IKBKB (0.44) PARP1FYNHSD17B1HSD17B2
SCHEMBL3165969 0.78 BAZ2B (0.44) PARP1DHODHBRD4NPC1RAB9A
SCHEMBL4916850 0.77 PARP1 (0.49) PARP1CHEK2ALDH1A1HSD17B10KDM4E
SCHEMBL4638595 0.77 HPGDS (0.46) PARP1CHEK2FYN
SCHEMBL731180 0.76 NQO2 (0.54) NQO2ALDH1A1NPC1RAB9ASMN1; SMN2
SCHEMBL694904 0.76 NQO2 (0.56) NQO2ALDH1A1NPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1991528-A2 MODULATORS OF ALPHA7 NICOTINIC ACETYLCHOLINE RECEPTORS AND THERAPEUTIC USES THEREOF Siena Biotech S.p.A. (IT) 2008-11-19 EP disclosed
WO-2007098826-A2 MODULATORS OF ALPHA7 NICOTINIC ACETYLCHOLINE RECEPTORS AND THERAPEUTIC USES THEREOF SIENA BIOTECH S.P.A. (IT) 2007-09-07 WO disclosed