SCHEMBL4655488

SCHEMBL4655488

CCC(Br)(NC(=O)OC(C)(C)C)C(=O)OC1CCCC1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 5/20 0.43
EPHX1 P07099 3/20 0.42
CYP19A1 P11511 1/20 0.38
GAA P10253 1/20 0.36
ALDH1A1 P00352 2/20 0.34
KMT2A Q03164 2/20 0.34
NAAA Q02083 2/20 0.34
BTK Q06187 1/20 0.34
MEN1 O00255 1/20 0.34
TSHR P16473 1/20 0.34
NPC1 O15118 1/20 0.33
HTT P42858 1/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
CTSS P25774 1/20 0.33
CTSK P43235 1/20 0.33
PDE4B Q07343 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4657733 0.99 EPHX1 (0.44) CACNA1BEPHX1CYP19A1GAAALDH1A1
SCHEMBL1151670 0.79 EPHX1 (0.41) CACNA1BEPHX1CYP19A1GAAKMT2A
SCHEMBL4628112 0.76 PTPRB (0.43) ALDH1A1KMT2AMEN1TSHRHTT
SCHEMBL2252759 0.75 EPHX1 (0.39) CACNA1BEPHX1CYP19A1GAAALDH1A1
SCHEMBL2252762 0.75 EPHX1 (0.39) CACNA1BEPHX1CYP19A1GAAALDH1A1
SCHEMBL29006969 0.71 BTK (0.36) CACNA1BEPHX1CYP19A1GAAALDH1A1
SCHEMBL26043772 0.71 EPHX1 (0.49) CACNA1BEPHX1CYP19A1GAABTK
SCHEMBL132134 0.70 EPHX1 (0.47) EPHX1CYP19A1NAAANPC1HTT
SCHEMBL12335551 0.70 EPHX1 (0.50) CACNA1BEPHX1GAAALDH1A1KMT2A
SCHEMBL25273708 0.69 KMT2A (0.48) CACNA1BEPHX1ALDH1A1KMT2ANAAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1877383-A1 QUINOLINE AND QUINOXALINE DERIVATIVES AS INHIBITORS OF KINASE ENZYMATIC ACTIVITY Chroma Therapeutics Limited (GB) 2008-01-16 EP disclosed
WO-2006117552-A1 QUINOLINE AND QUINOXALINE DERIVATIVES AS INHIBITORS OF KINASE ENZYMATIC ACTIVITY CHROMA THERAPEUTICS LTD (GB) 2006-11-09 WO disclosed