SCHEMBL4655682

SCHEMBL4655682

O=C(NC1CCCC(O)(C#Cc2cccc(Cl)c2)C1)c1ccc(F)c(F)c1

nearest known ligand 0.48

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 15/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
TAS1R3 Q7RTX0 1/20 0.40
TAS1R1 Q7RTX1 1/20 0.40
TAS1R2 Q8TE23 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL990824 1.00 GRM5 (0.48) GRM5L3MBTL1NPC1RAB9AMEN1
SCHEMBL992253 1.00 GRM5 (0.48) GRM5L3MBTL1NPC1RAB9AMEN1
SCHEMBL990340 0.91 L3MBTL1 (0.59) GRM5L3MBTL1NPC1RAB9AMEN1
SCHEMBL990772 0.90 GRM5 (0.60) GRM5L3MBTL1NPC1RAB9AMEN1
SCHEMBL3799474 0.90 GRM5 (0.47) GRM5L3MBTL1NPC1RAB9A
2-Picolinic Acid SCHEMBL3631655 0.89 GRM5 (0.50) GRM5L3MBTL1
SCHEMBL2818567 0.88 L3MBTL1 (0.47) GRM5L3MBTL1NPC1RAB9AMEN1
SCHEMBL992266 0.87 L3MBTL1 (0.46) GRM5L3MBTL1NPC1RAB9AMEN1
SCHEMBL990869 0.87 GRM5 (0.48) GRM5L3MBTL1NPC1RAB9AMEN1
SCHEMBL990083 0.87 L3MBTL1 (0.47) GRM5L3MBTL1NPC1RAB9AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1877365-A1 ACETYLENE DERIVATIVES Novartis AG (CH) 2008-01-16 EP disclosed
WO-2006114262-A1 ACETYLENE DERIVATIVES NOVARTIS AG (CH) 2006-11-02 WO disclosed