SCHEMBL4656555

SCHEMBL4656555

NC(=O)Oc1sc2nc(N3CCC(N)CC3)cc(C(F)(F)F)c2c1N

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 1/20 0.52
TMEM97 Q5BJF2 1/20 0.52
IKBKB O14920 15/20 0.48
CHUK O15111 2/20 0.48
EPHA3 P29320 2/20 0.48
GAK O14976 1/20 0.47
ICAM1 P05362 1/20 0.47
DRD2 P14416 1/20 0.47
NFKBIA P25963 1/20 0.47
DRD3 P35462 1/20 0.47
ABAT P80404 1/20 0.47
AAK1 Q2M2I8 1/20 0.47
IRAK3 Q9Y616 1/20 0.47
MEN1 O00255 2/20 0.41
ALDH1A1 P00352 2/20 0.41
HPGD P15428 2/20 0.41
KMT2A Q03164 2/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
NTRK1 P04629 1/20 0.39
KDM4E B2RXH2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4657007 0.92 SLC6A3 (0.52) SLC6A3TMEM97IKBKBCHUKEPHA3
SCHEMBL4659135 0.87 IKBKB (0.51) SLC6A3TMEM97IKBKBCHUKEPHA3
SCHEMBL4657084 0.85 IKBKB (0.66) SLC6A3TMEM97IKBKBCHUKEPHA3
SCHEMBL4657748 0.82 IKBKB (0.50) IKBKBCHUKEPHA3GAKICAM1
SCHEMBL4657934 0.80 IKBKB (0.53) IKBKBCHUKEPHA3GAKICAM1
SCHEMBL4657206 0.79 IKBKB (0.44) SLC6A3TMEM97IKBKBCHUKEPHA3
SCHEMBL4659402 0.79 IKBKB (0.44) IKBKBCHUKEPHA3GAKICAM1
SCHEMBL4657927 0.79 IKBKB (0.44) IKBKBCHUKEPHA3GAKICAM1
SCHEMBL4656552 0.78 IKBKB (0.45) SLC6A3TMEM97IKBKBCHUKEPHA3
SCHEMBL4656940 0.78 IKBKB (0.69) IKBKBCHUKEPHA3NTRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1513516-B1 SUBSTITUTED 3-AMINO-THIENO(2,3-b) PYRIDINE-2-CARBOXYLIC ACID AMIDE COMPOUNDS AND PROCESSES FOR PREPARING AND THEIR USES BOEHRINGER INGELHEIM PHARMA (US) 2008-12-03 EP claimed