Vigabatrin

Vigabatrin

SCHEMBL465981

C=C[C@@H](N)CCC(=O)O

nearest known ligand 0.00

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABAT

The experimentally established mechanism targets of Vigabatrin. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Vigabatrin SCHEMBL9132153 1.00
Vigabatrin SCHEMBL5785801 1.00 CYP2D6 (1.00)
Vigabatrin SCHEMBL26714 1.00
Vigabatrin SCHEMBL31159534 1.00
Vigabatrin SCHEMBL20659806 0.98 CYP2D6 (0.95)
Vigabatrin SCHEMBL17372729 0.88 BLM (0.78)
Valproic Acid SCHEMBL2372220 0.84 SLC6A3 (0.70)
Hydrochloric Acid SCHEMBL31483557 0.79 BLM (0.65)
SCHEMBL15396442 0.79
SCHEMBL8058851 0.79

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 773 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3607938-B1 PHARMACEUTICAL COMPOSITION SOVIC BRKICIC LJILJANA (HR) 2026-05-27 EP claimed
EP-4181891-B1 USE OF CANNABIDIOL IN THE TREATMENT OF ABSENCE SEIZURES ASSOCIATED WITH RARE EPILEPSY SYNDROMES RELATED TO BRAIN INJURY JAZZ PHARMACEUTICALS RESEARCH UK LTD (GB) 2025-12-17 EP claimed
EP-4043016-B1 THE 5HT AGONIST CLEMIZOLE FOR USE IN TREATING EPILEPSY DISORDERS UNIV CALIFORNIA (US) 2025-10-29 EP claimed
EP-4181901-B1 USE OF CANNABIDIOL IN THE TREATMENT OF SEIZURES ASSOCIATED WITH RARE EPILEPSY SYNDROMES RELATED TO GENETIC ABNORMALITIES JAZZ PHARMACEUTICALS RESEARCH UK LTD (GB) 2025-10-15 EP claimed
EP-3436000-B1 USE OF CANNABINOIDS IN THE TREATMENT OF STURGE WEBER SYNDROME JAZZ PHARMACEUTICALS RESEARCH UK LTD (GB) 2025-07-16 EP claimed
EP-3917907-B1 MODULATORS OF POTASSIUM ION CHANNELS AND USES THEREOF UNIV DEGLI STUDI DI SALERNO (IT) 2025-05-21 EP claimed
EP-4181899-B1 USE OF CANNABIDIOL IN THE TREATMENT OF SEIZURES ASSOCIATED WITH RARE EPILEPSY SYNDROMES RELATED TO GENETIC ABNORMALITIES JAZZ PHARMACEUTICALS RESEARCH UK LTD (GB) 2025-05-21 EP claimed
EP-3518975-B1 FORMULATION COMPRISING FENFLURAMINE AND CANNABIDIOL AND ITS USE IN THE TREATMENT OF SEIZURES ZOGENIX INTERNATIONAL LTD (GB) 2025-04-09 EP claimed
EP-3638673-B9 TETRAHYDROPYRIDOPYRAZINE MODULATORS OF GPR6 TAKEDA PHARMACEUTICALS CO (JP) 2024-11-20 EP claimed
EP-3615010-B1 METHODS FOR TREATING DRAVET SYNDROME CAVION INC (US) 2024-08-21 EP claimed
EP-1438019-A1 KIT FOR THE PREPARATION OF A PHARMACEUTICAL COMPOSITION PARI GmbH Spezialisten für effektive Inhalation (DE) 2004-07-21 EP claimed
EP-0956019-B1 NOVEL THERAPEUTIC APPLICATION OF A THIENYCYCLOHEXYLAMINE DERIVATIVE SOD CONSEILS RECH APPLIC (FR) 2003-10-15 EP claimed
WO-2003035030-A1 KIT FOR THE PREPARATION OF A PHARMACEUTICAL COMPOSITION PARI GMBH (DE) 2003-05-01 WO claimed
WO-2003000643-A1 NITRATE ESTER DERIVATIVES USEFUL FOR PREPARING DRUGS FOR EPILEPSY NICOX S.A. (FR) 2003-01-03 WO claimed
EP-1227856-A1 INHALATION NEBULIZER PARI GmbH Spezialisten für effektive Inhalation (DE) 2002-08-07 EP claimed
WO-2001034232-A9 INHALATION NEBULIZER PARI GMBH (DE) 2002-08-01 WO claimed
WO-2001034232-A1 INHALATION NEBULIZER Pari GmbH Spezialisten für effektive Inhalation (DE) 2001-05-17 WO claimed
EP-0956019-A1 NOVEL THERAPEUTIC APPLICATION OF A THIENYCYCLOHEXYLAMINE DERIVATIVE SOCIETE DE CONSEILS DE RECHERCHES ET D'APPLICATIONS SCIENTIFIQUES (S.C.R.A.S.) (FR) 1999-11-17 EP claimed
WO-1998024434-A1 NOVEL THERAPEUTIC APPLICATION OF A THIENYCYCLOHEXYLAMINE DERIVATIVE SOCIETE DE CONSEILS DE RECHERCHES ET D'APPLICATIONS SCIENTIFIQUES (S.C.R.A.S.) (FR) 1998-06-11 WO claimed
EP-0463560-B1 New antiepileptic agents CIBA GEIGY AG (CH) 1995-10-25 EP claimed