SCHEMBL4661297

SCHEMBL4661297

CC(C)(C)NC(=O)CCc1ccc(CNc2c(Cl)ccc3c2CCCCN3)cc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
MAPT P10636 3/20 0.35
PARP1 P09874 3/20 0.33
ALDH1A1 P00352 3/20 0.33
PRCP P42785 1/20 0.33
FFAR1 O14842 2/20 0.33
CDK1 P06493 1/20 0.32
CDK2 P24941 1/20 0.32
MAPK1 P28482 1/20 0.32
GSK3A P49840 1/20 0.32
GSK3B P49841 1/20 0.32
P2RX7 Q99572 2/20 0.32
ANO1 Q5XXA6 1/20 0.32
KDM4E B2RXH2 1/20 0.32
MEN1 O00255 1/20 0.32
GAA P10253 1/20 0.32
G6PD P11413 1/20 0.32
HPGD P15428 1/20 0.32
BLM P54132 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2584431 0.81 HTR2A (0.37) CA1CA2MAPTALDH1A1PRCP
Cadaverine Tartrate SCHEMBL13685478 0.76 FFAR1 (0.33) CA1CA2MAPTALDH1A1PRCP
SCHEMBL2586609 0.75 POLB (0.34) PARP1ALDH1A1CDK1CDK2MAPK1
Succinic Acid SCHEMBL5729110 0.74 FFAR1 (0.32) FFAR1KDM4EMEN1HPGDKMT2A
Succinic Acid SCHEMBL5735783 0.73 HPGD (0.33) PARP1ALDH1A1FFAR1KDM4EHPGD
SCHEMBL2581859 0.73 ESR1 (0.37) CA1CA2MAPTALDH1A1FFAR1
Succinic Acid SCHEMBL5757273 0.72 HRH3 (0.36) PARP1ALDH1A1FFAR1HPGD
SCHEMBL2584611 0.70 HTR2A (0.36) ALDH1A1FFAR1P2RX7MEN1KMT2A
SCHEMBL4774872 0.70 P2RX3 (0.30)
SCHEMBL507619 0.69 HTR2A (0.39) FFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1924561-A2 6-ARYLALKYLAMINO- 2,3,4,5-TETRAHYDRO-1H-BENZO[D]AZEPINES AS 5-HT2C RECEPTOR AGONISTS Eli Lilly & Company (US) 2008-05-28 EP disclosed
WO-2007028083-A2 6-ARYLALKYLAMINO- 2,3,4,5-TETRAHYDRO-1H-BENZO[D]AZEPINES AS 5-HT2C RECEPTOR AGONISTS ELI LILLY AND COMPANY (US) 2007-03-08 WO disclosed