SCHEMBL4661576

SCHEMBL4661576

CC(C)(C)OC(=O)C(C)(C#N)C(c1ccccc1C(F)(F)F)c1cccc2ccccc12

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.45
ESR2 Q92731 1/20 0.45
SLC6A4 P31645 1/20 0.38
KDM4E B2RXH2 2/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
CTSS P25774 1/20 0.37
CTSK P43235 1/20 0.37
HDAC3 O15379 1/20 0.35
CYP2C9 P11712 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
AR P10275 1/20 0.35
LMNA P02545 2/20 0.34
POLB P06746 1/20 0.34
CNR2 P34972 2/20 0.33
GAA P10253 1/20 0.32
ALDH1A1 P00352 1/20 0.32
HSD17B10 Q99714 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4660033 0.86 ESR1 (0.46) ESR1ESR2SLC6A4KDM4EMEN1
SCHEMBL4661381 0.85 ESR1 (0.41) ESR1ESR2KDM4EMEN1KMT2A
SCHEMBL4660073 0.85 ESR1 (0.41) ESR1ESR2KDM4EMEN1KMT2A
SCHEMBL4660190 0.85 ESR1 (0.48) ESR1ESR2KDM4EMEN1KMT2A
SCHEMBL4661489 0.84 ESR1 (0.53) ESR1ESR2SLC6A4KDM4EMEN1
SCHEMBL4662659 0.84 ESR1 (0.53) ESR1ESR2SLC6A4KDM4EMEN1
SCHEMBL4661552 0.82 ESR1 (0.39) ESR1ESR2KDM4EMEN1KMT2A
SCHEMBL4661562 0.77 ESR1 (0.43) ESR1ESR2KDM4EKMT2ACNR2
SCHEMBL4661384 0.76 SLC6A4 (0.38) ESR1ESR2SLC6A4KDM4EMEN1
SCHEMBL4135203 0.75 ESR1 (0.54) ESR1ESR2SLC6A4KDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1620102-B1 3-(1-NAPHTHYL)-2-CYANOPROPANOIC ACID DERIVATIVES AS ESTROGEN RECEPTOR LIGANDS WYETH CORP (US) 2008-12-24 EP claimed