Pyrrole

Pyrrole

SCHEMBL4661864

O=C(O)c1cccc2cc[nH]c12.c1cc[nH]c1

nearest known ligand 0.86

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.86
PDPK1 O15530 1/20 0.62
GRM5 P41594 1/20 0.47
BACE1 P56817 1/20 0.46
HDAC1 Q13547 3/20 0.46
HDAC2 Q92769 3/20 0.46
HDAC3 O15379 2/20 0.46
HDAC4 P56524 2/20 0.46
HDAC7 Q8WUI4 2/20 0.46
HDAC10 Q969S8 2/20 0.46
HDAC11 Q96DB2 2/20 0.46
HDAC8 Q9BY41 2/20 0.46
HDAC6 Q9UBN7 2/20 0.46
HDAC9 Q9UKV0 2/20 0.46
HDAC5 Q9UQL6 2/20 0.46
NR4A1 P22736 1/20 0.43
NR4A2 P43354 1/20 0.43
NR4A3 Q92570 1/20 0.43
AHR P35869 1/20 0.43
MAPT P10636 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29696550 0.93 KEAP1 (1.00) KEAP1PDPK1GRM5BACE1HDAC1
SCHEMBL336234 0.93 KEAP1 (1.00) KEAP1PDPK1GRM5BACE1HDAC1
Hydrochloric Acid SCHEMBL8595147 0.91 KEAP1 (0.96) KEAP1PDPK1GRM5BACE1HDAC1
SCHEMBL4719779 0.81 KEAP1 (0.76) KEAP1PDPK1GRM5BACE1HDAC1
SCHEMBL888364 0.77 KEAP1 (0.64) KEAP1PDPK1GRM5BACE1HDAC1
SCHEMBL27967849 0.77 KEAP1 (0.70) KEAP1PDPK1GRM5BACE1HDAC1
SCHEMBL1651352 0.77 PDPK1 (1.00) KEAP1PDPK1GRM5BACE1HDAC1
SCHEMBL29567411 0.77 PDPK1 (1.00) KEAP1PDPK1GRM5BACE1HDAC1
SCHEMBL30690400 0.77 KEAP1 (0.70) KEAP1PDPK1GRM5BACE1HDAC1
SCHEMBL27968063 0.77 KEAP1 (0.70) KEAP1PDPK1GRM5BACE1HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0819133-B1 COVALENTLY LINKED OLIGONUCLEOTIDE MINOR GROOVE BINDER CONJUGATES EPOCH BIOSCIENCES INC (US) 2008-01-02 EP disclosed