SCHEMBL4662273

SCHEMBL4662273

CN1C(=O)NC(=O)C12Cc1ccc([AsH2])cc1C2

nearest known ligand 0.43

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CALCRL Q16602 19/20 0.43
MAP2K2 P36507 1/20 0.41
ADM2 Q7Z4H4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12921079 0.83 BRD4 (0.46) CALCRLMAP2K2
SCHEMBL1921018 0.83 BRD4 (0.46) CALCRLMAP2K2
SCHEMBL16624586 0.83 CALCRL (0.53) CALCRLMAP2K2
SCHEMBL13192493 0.81 CALCRL (0.43) CALCRLMAP2K2ADM2
SCHEMBL378986 0.81 CALCRL (0.46) CALCRLMAP2K2
SCHEMBL1394328 0.81 CALCRL (0.46) CALCRLMAP2K2
SCHEMBL1274913 0.81 CALCRL (0.46) CALCRLMAP2K2
SCHEMBL15401458 0.78 CALCRL (0.46) CALCRLMAP2K2ADM2
SCHEMBL1394805 0.78 TDP2 (0.47) CALCRL
SCHEMBL15400764 0.78 CALCRL (0.46) CALCRLMAP2K2ADM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1608627-B1 BICYCLIC ANILIDE SPIROHYDANTOIN CGRP RECEPTOR ANTAGONISTS MERCK & CO INC (US) 2008-05-07 EP disclosed