SCHEMBL4666895

SCHEMBL4666895

FC(F)(F)c1ccc(C23C[C@H]2CN(CCCCl)C3)nc1

nearest known ligand 0.45

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 17/20 0.45
KCNH2 Q12809 16/20 0.45
DRD2 P14416 14/20 0.45
CYP1A2 P05177 1/20 0.42
DRD4 P21917 1/20 0.40
CYP2C19 P33261 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3555050 1.00 DRD3 (0.45) DRD3KCNH2DRD2CYP1A2DRD4
SCHEMBL13312904 1.00 DRD3 (0.45) DRD3KCNH2DRD2CYP1A2DRD4
SCHEMBL3623998 1.00 DRD3 (0.45) DRD3KCNH2DRD2CYP1A2DRD4
SCHEMBL12809870 0.90 DRD3 (0.44) DRD3KCNH2DRD2CYP1A2DRD4
SCHEMBL14567571 0.90 DRD3 (0.44) DRD3KCNH2DRD2CYP1A2DRD4
SCHEMBL378256 0.83 DRD3 (0.55) DRD3KCNH2DRD2CYP1A2
SCHEMBL13089084 0.83 DRD3 (0.55) DRD3KCNH2DRD2CYP1A2
SCHEMBL379237 0.83 POLB (0.41) DRD3KCNH2DRD2
SCHEMBL12313188 0.83 POLB (0.41) DRD3KCNH2DRD2
SCHEMBL11911752 0.83 POLB (0.41) DRD3KCNH2DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1926723-A2 AZABICYCLO (3,1,0) HEXAN DERIVATIVES USEFUL AS MODULATORS OF DOPAMINE D3 RCEPTORS GLAXO GROUP LIMITED (GB) 2008-06-04 EP disclosed
WO-2007022934-A2 AZABICYCLO (3, 1, 0) HEXAN DERIVATIVES USEFUL AS MODULATORS OF DOPAMINE D3 RECEPTORS GLAXO GROUP LIMITED (GB) 2007-03-01 WO disclosed