SCHEMBL4667840

SCHEMBL4667840

COc1c(-c2ccccc2)nc2ccccc2c1C(=O)N[C@@H](C)c1ccccc1C#N

nearest known ligand 0.59

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 20/20 0.59
TACR2 P21452 3/20 0.59
CYP3A4 P08684 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4665574 0.87 TACR3 (0.57) TACR3TACR2CYP3A4
SCHEMBL4667323 0.87 TACR3 (0.57) TACR3TACR2CYP3A4
SCHEMBL4668719 0.87 TACR3 (0.57) TACR3TACR2
SCHEMBL4665598 0.84 TACR3 (0.50) TACR3TACR2
SCHEMBL4665564 0.82 TACR3 (0.61) TACR3TACR2CYP3A4
SCHEMBL5042628 0.82 TACR3 (0.62) TACR3TACR2
SCHEMBL14094523 0.79 TACR3 (0.62) TACR3TACR2CYP3A4
SCHEMBL4667842 0.78 TACR3 (0.56) TACR3TACR2CYP3A4
SCHEMBL4667841 0.77 TACR3 (0.78) TACR3TACR2CYP3A4
SCHEMBL14015208 0.77 TACR3 (0.59) TACR3TACR2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1928834-A1 ALKYLNITRILE QUINOLINES, AS NK-3 RECEPTOR LIGANDS AstraZeneca AB (SE) 2008-06-11 EP claimed
WO-2007035157-A1 ALKYLNITRILE QUINOLINES, AS NK-3 RECEPTOR LIGANDS ASTRAZENECA AB (SE) 2007-03-29 WO claimed
EP-1928834-A1 ALKYLNITRILE QUINOLINES, AS NK-3 RECEPTOR LIGANDS AstraZeneca AB (SE) 2008-06-11 EP disclosed
WO-2007035157-A1 ALKYLNITRILE QUINOLINES, AS NK-3 RECEPTOR LIGANDS ASTRAZENECA AB (SE) 2007-03-29 WO disclosed