SCHEMBL4668374

SCHEMBL4668374

NC(=O)Nc1cc(Cl)ccc1OCC(=O)NC1CC2CCC(C1)N2Cc1ccc(Cl)cc1.NC(=O)c1cc(Cl)ccc1OCC(=O)NC1CC2CCC(C1)N2Cc1ccc(Cl)cc1

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.47
RAB9A P51151 2/20 0.47
CCR1 P32246 2/20 0.44
FPR3 P25089 1/20 0.44
GPR65 Q8IYL9 1/20 0.44
GPR35 Q9HC97 1/20 0.44
MCHR1 Q99705 1/20 0.44
CXCR6 O00574 1/20 0.43
MAPT P10636 1/20 0.42
MAPK1 P28482 1/20 0.42
LMNA P02545 1/20 0.42
HPGD P15428 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
OPRK1 P41145 1/20 0.41
KCNH2 Q12809 1/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
NPSR1 Q6W5P4 1/20 0.41
DRD2 P14416 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4668370 1.00 NPC1 (0.47) NPC1RAB9ACCR1FPR3GPR65
SCHEMBL3869168 0.95 CCR1 (0.48) NPC1RAB9ACCR1FPR3GPR65
SCHEMBL3869170 0.95 CCR1 (0.48) NPC1RAB9ACCR1FPR3GPR65
SCHEMBL3869555 0.95 CCR1 (0.48) NPC1RAB9ACCR1FPR3GPR65
SCHEMBL3873444 0.93 NPC1 (0.53) NPC1RAB9AMCHR1CXCR6LMNA
SCHEMBL3873441 0.93 NPC1 (0.53) NPC1RAB9AMCHR1CXCR6LMNA
SCHEMBL4669557 0.91 CCR1 (0.45) NPC1RAB9ACCR1FPR3GPR65
SCHEMBL4669555 0.91 CCR1 (0.45) NPC1RAB9ACCR1FPR3GPR65
SCHEMBL13853100 0.90 MCHR1 (0.54) NPC1CCR1FPR3GPR65GPR35
SCHEMBL3869061 0.90 CCR1 (0.55) NPC1RAB9ACCR1FPR3GPR65

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1891064-A1 N-AMIDE DERIVATIVES OF 8-AZABICYCLO[3.2.1]OCT-3-YL AS CCR1 ANTAGONISTS Laboratorios Almirall, S.A. (ES) 2008-02-27 EP claimed
WO-2006133802-A1 N-AMIDE DERIVATIVES OF 8-AZABICYCLO[3.2.1]OCT-3-YL AS CCR1 ANTAGONISTS LABORATORIOS ALMIRALL, S.A. (ES) 2006-12-21 WO claimed
EP-1891064-A1 N-AMIDE DERIVATIVES OF 8-AZABICYCLO[3.2.1]OCT-3-YL AS CCR1 ANTAGONISTS Laboratorios Almirall, S.A. (ES) 2008-02-27 EP disclosed
WO-2006133802-A1 N-AMIDE DERIVATIVES OF 8-AZABICYCLO[3.2.1]OCT-3-YL AS CCR1 ANTAGONISTS LABORATORIOS ALMIRALL, S.A. (ES) 2006-12-21 WO disclosed