SCHEMBL4669557

SCHEMBL4669557

N=C(N)Nc1cc(Cl)ccc1OCC(=O)NC1CC2CCC(C1)N2Cc1ccc(Cl)cc1.NC(=O)Nc1cc(Cl)ccc1OCC(=O)NC1CC2CCC(C1)N2Cc1ccc(Cl)cc1

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 2/20 0.45
FPR3 P25089 1/20 0.45
GPR65 Q8IYL9 1/20 0.45
GPR35 Q9HC97 1/20 0.45
MCHR1 Q99705 1/20 0.45
CXCR6 O00574 1/20 0.44
NPC1 O15118 4/20 0.44
MAPT P10636 1/20 0.43
MAPK1 P28482 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
LMNA P02545 1/20 0.43
HPGD P15428 1/20 0.43
RAB9A P51151 3/20 0.41
KMT2A Q03164 2/20 0.40
MEN1 O00255 1/20 0.40
LTA4H P09960 1/20 0.40
ALDH1A1 P00352 1/20 0.40
ACHE P22303 1/20 0.39
ATF4 P18848 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4669555 1.00 CCR1 (0.45) CCR1FPR3GPR65GPR35MCHR1
SCHEMBL3871383 0.97 NPC1 (0.46) CCR1FPR3GPR65GPR35MCHR1
SCHEMBL3871382 0.97 NPC1 (0.46) CCR1FPR3GPR65GPR35MCHR1
SCHEMBL3869168 0.96 CCR1 (0.48) CCR1FPR3GPR65GPR35MCHR1
SCHEMBL3869170 0.96 CCR1 (0.48) CCR1FPR3GPR65GPR35MCHR1
SCHEMBL3869555 0.96 CCR1 (0.48) CCR1FPR3GPR65GPR35MCHR1
SCHEMBL13853100 0.91 MCHR1 (0.54) CCR1FPR3GPR65GPR35MCHR1
SCHEMBL4668370 0.91 NPC1 (0.47) CCR1FPR3GPR65GPR35MCHR1
SCHEMBL4668374 0.91 NPC1 (0.47) CCR1FPR3GPR65GPR35MCHR1
SCHEMBL3869061 0.90 CCR1 (0.55) CCR1FPR3GPR65GPR35MCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1891064-A1 N-AMIDE DERIVATIVES OF 8-AZABICYCLO[3.2.1]OCT-3-YL AS CCR1 ANTAGONISTS Laboratorios Almirall, S.A. (ES) 2008-02-27 EP claimed
WO-2006133802-A1 N-AMIDE DERIVATIVES OF 8-AZABICYCLO[3.2.1]OCT-3-YL AS CCR1 ANTAGONISTS LABORATORIOS ALMIRALL, S.A. (ES) 2006-12-21 WO claimed