SCHEMBL4669307

SCHEMBL4669307

COc1ccc(C#N)cc1C#N.N#Cc1ccc(O)c(C#N)c1

nearest known ligand 0.53

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.53
KDM4E B2RXH2 1/20 0.53
USP2 O75604 1/20 0.53
AR P10275 9/20 0.47
PGR P06401 1/20 0.47
IMPDH2 P12268 1/20 0.45
IMPDH1 P20839 1/20 0.45
ESRRA P11474 1/20 0.42
P4HB P07237 2/20 0.40
EGFR P00533 1/20 0.40
GUSB P08236 1/20 0.39
DYRK1A Q13627 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2094284 0.89 ALDH1A1 (0.63) ALDH1A1KDM4EUSP2ARIMPDH2
SCHEMBL2635720 0.84 CA12 (0.48) ARIMPDH2IMPDH1
SCHEMBL29804271 0.80 MAOB (0.55) ALDH1A1ARP4HBEGFRGUSB
SCHEMBL459931 0.80 MAOB (0.55) ALDH1A1ARP4HBEGFRGUSB
SCHEMBL388024 0.80 AR (0.51) ALDH1A1ARP4HB
Methyl Alcohol SCHEMBL27451617 0.79 AR (0.50) ALDH1A1ARP4HB
SCHEMBL24476682 0.78 AR (0.54) ALDH1A1KDM4EUSP2ARPGR
SCHEMBL2793117 0.77 ALDH1A1 (0.58) ALDH1A1KDM4EUSP2ARIMPDH2
SCHEMBL16951586 0.77 AR (0.49) ALDH1A1KDM4EUSP2ARIMPDH2
SCHEMBL16950438 0.77 ALDH1A1 (0.58) ALDH1A1KDM4EUSP2ARPGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1893619-A1 NEW OXABISPIDINE COMPOUNDS FOR THE TREATMENT OF CARDIAC ARRHYTMIAS AstraZeneca AB (SE) 2008-03-05 EP disclosed
WO-2006135316-A1 New oxabispidine compounds for the treatment of cardiac arrhythmias ASTRAZENECA AB (SE) 2006-12-21 WO disclosed