SCHEMBL4675392

SCHEMBL4675392

c1cncc(CNN2CCCC2)c1

nearest known ligand 0.57

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.57
CHRNA4 P43681 1/20 0.57
CYP1A2 P05177 1/20 0.56
CYP2D6 P10635 1/20 0.56
ALDH1A1 P00352 4/20 0.51
KDM4E B2RXH2 1/20 0.51
PKM P14618 1/20 0.51
HSD17B10 Q99714 2/20 0.49
LTA4H P09960 1/20 0.49
CHRM2 P08172 1/20 0.47
KDM1A O60341 2/20 0.47
MAOA P21397 1/20 0.47
MAOB P27338 1/20 0.47
NPSR1 Q6W5P4 1/20 0.46
RECQL P46063 1/20 0.46
NAMPT P43490 1/20 0.46
CYP2C19 P33261 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10512212 0.85 CHRNB2 (0.43) CHRNB2CHRNA4CYP1A2CYP2D6ALDH1A1
SCHEMBL10512608 0.84 NAMPT (0.44) CHRNB2CHRNA4CYP1A2CYP2D6ALDH1A1
SCHEMBL2255128 0.77 DPP7 (0.52) ALDH1A1KDM4E
SCHEMBL518257 0.76 DPP7 (0.50) CYP1A2CYP2D6ALDH1A1KDM4ECYP2C19
SCHEMBL8522936 0.75 CYP1A2 (0.60) CYP1A2CYP2D6ALDH1A1KDM4EPKM
SCHEMBL10512848 0.74 MAPT (0.48) CYP1A2CYP2D6ALDH1A1NAMPTCYP2C19
SCHEMBL8647480 0.74 DPP7 (0.47) ALDH1A1KDM4EKDM1AMAOA
SCHEMBL6538443 0.73 DPP7 (0.65) CHRNB2CHRNA4CYP1A2CYP2D6ALDH1A1
SCHEMBL5361875 0.73 CYP1A2 (0.75) CYP1A2CYP2D6ALDH1A1KDM4EPKM
SCHEMBL2861457 0.73 CYP1A2 (1.00) CYP1A2CYP2D6ALDH1A1LTA4HCHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1951689-A1 P2X7 RECEPTOR ANTAGONISTS AND METHODS OF USE ABBOTT LABORATORIES (US) 2008-08-06 EP disclosed
WO-2007056046-A1 P2X7 RECEPTOR ANTAGONISTS AND METHODS OF USE ABBOTT LABORATORIES (US) 2007-05-18 WO disclosed