SCHEMBL4676331

SCHEMBL4676331

C[C@H](N)C(=O)NNC(=O)NCc1ccc(F)cc1

nearest known ligand 0.55

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.55
TSHR P16473 1/20 0.55
ANPEP P15144 1/20 0.54
HPGD P15428 2/20 0.54
GAA P10253 3/20 0.52
MEN1 O00255 3/20 0.52
KMT2A Q03164 3/20 0.52
CARM1 Q86X55 2/20 0.50
PRMT6 Q96LA8 2/20 0.50
L3MBTL1 Q9Y468 1/20 0.49
RAB9A P51151 3/20 0.49
POLB P06746 2/20 0.49
NPC1 O15118 1/20 0.49
MAOB P27338 1/20 0.49
ALDH1A1 P00352 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4680706 1.00 MAPK1 (0.55) MAPK1TSHRANPEPHPGDGAA
SCHEMBL10692282 0.86 CARM1 (0.62) MAPK1TSHRANPEPHPGDGAA
SCHEMBL4677304 0.85 MEN1 (0.60) TSHRHPGDMEN1KMT2ACARM1
SCHEMBL4677340 0.85 MEN1 (0.60) TSHRHPGDMEN1KMT2ACARM1
SCHEMBL4676692 0.85 SMN1; SMN2 (0.53) ANPEPGAAMEN1KMT2AL3MBTL1
SCHEMBL4676219 0.85 SMN1; SMN2 (0.53) ANPEPGAAMEN1KMT2AL3MBTL1
Hydrochloric Acid SCHEMBL5967401 0.84 CARM1 (0.64) MAPK1TSHRANPEPHPGDGAA
SCHEMBL4679395 0.83 ANPEP (0.58) MAPK1ANPEPCARM1PRMT6RAB9A
SCHEMBL4676327 0.83 ANPEP (0.58) MAPK1ANPEPCARM1PRMT6RAB9A
SCHEMBL8302088 0.80 ERCC1 (0.62) CARM1PRMT6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1633702-B1 PROTEASE INHIBITORS PROZYMEX AS (DK) 2008-07-02 EP claimed
US-20070155803-A1 Protease inhibitors PROZYMEX A/S (DK) 2007-07-05 US claimed
EP-1633702-A1 PROTEASE INHIBITORS Prozymex A/S (DK) 2006-03-15 EP claimed
WO-2004106289-A1 PROTEASE INHIBITORS PROZYMEX A/S (DK) 2004-12-09 WO claimed
EP-1975153-A2 Protease inhibitors Prozymex A/S (DK) 2008-10-01 EP disclosed
EP-1975153-A2 Protease inhibitors Prozymex A/S (DK) 2008-10-01 EP disclosed
EP-1633702-B1 PROTEASE INHIBITORS PROZYMEX AS (DK) 2008-07-02 EP disclosed
US-20070155803-A1 Protease inhibitors PROZYMEX A/S (DK) 2007-07-05 US disclosed
US-20070155803-A1 Protease inhibitors PROZYMEX A/S (DK) 2007-07-05 US disclosed
US-20070155803-A1 Protease inhibitors PROZYMEX A/S (DK) 2007-07-05 US disclosed
EP-1633702-A1 PROTEASE INHIBITORS Prozymex A/S (DK) 2006-03-15 EP disclosed
WO-2004106289-A1 PROTEASE INHIBITORS PROZYMEX A/S (DK) 2004-12-09 WO disclosed
WO-2004106289-A1 PROTEASE INHIBITORS PROZYMEX A/S (DK) 2004-12-09 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070155803-A1 Protease inhibitors DPP7, DPP9, DPP3 MAPK1 4154/4885TSHR 2862/4885ANPEP 112/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.