SCHEMBL4677495

SCHEMBL4677495

COc1cccc(C=C2OC(=O)c3ccccc32)c1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.61
HPGD P15428 7/20 0.61
KDM4E B2RXH2 5/20 0.61
L3MBTL1 Q9Y468 3/20 0.61
TDP1 Q9NUW8 1/20 0.61
MEN1 O00255 5/20 0.59
KMT2A Q03164 5/20 0.59
MAPT P10636 4/20 0.59
CYP1A2 P05177 3/20 0.55
CYP2C19 P33261 3/20 0.55
SMN1; SMN2 Q16637 3/20 0.55
CYP3A4 P08684 2/20 0.55
POLB P06746 1/20 0.55
CYP2C9 P11712 1/20 0.55
NFKB1 P19838 1/20 0.55
NFKB2 Q00653 1/20 0.55
RELA Q04206 1/20 0.55
NPC1 O15118 3/20 0.53
RAB9A P51151 3/20 0.53
PKM P14618 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11176235 1.00 ALDH1A1 (0.61) ALDH1A1HPGDKDM4EL3MBTL1TDP1
SCHEMBL4677493 1.00 ALDH1A1 (0.61) ALDH1A1HPGDKDM4EL3MBTL1TDP1
SCHEMBL22259113 0.86 MAPT (0.59) ALDH1A1HPGDKDM4EL3MBTL1MEN1
SCHEMBL2820796 0.83 KDM4E (0.69) ALDH1A1HPGDKDM4EL3MBTL1TDP1
SCHEMBL2820798 0.83 KDM4E (0.69) ALDH1A1HPGDKDM4EL3MBTL1TDP1
SCHEMBL28572859 0.82 KDM4E (0.61) ALDH1A1HPGDKDM4EL3MBTL1TDP1
SCHEMBL30395765 0.82 KDM4E (0.61) ALDH1A1HPGDKDM4EL3MBTL1TDP1
SCHEMBL28996362 0.82 KDM4E (0.61) ALDH1A1HPGDKDM4EL3MBTL1TDP1
SCHEMBL9764623 0.80 ALDH1A1 (0.69) ALDH1A1HPGDKDM4EL3MBTL1TDP1
SCHEMBL29637242 0.80 ALDH1A1 (0.69) ALDH1A1HPGDKDM4EL3MBTL1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4333920-A Benzalphthalides and broad spectrum sun screens VAN DYK & COMPANY, INC. (US) 1982-06-08 US claimed
CN-108752300-B Benzylidene phenylene peptide compound, pharmaceutical composition and application thereof 中国科学院昆明植物研究所 2022-03-25 CN disclosed
CN-108752300-A Benzyl alkene pitches benzene peptides and its pharmaceutical composition and its application 中国科学院昆明植物研究所 2018-11-06 CN disclosed
EP-1216994-B1 Tricyclic antidepressant derivatives and immunoassay ROCHE DIAGNOSTICS GMBH (DE) 2008-12-31 EP disclosed
EP-1216994-A2 Tricyclic antidepressant derivatives and immunoassay Roche Diagnostics GmbH (DE) 2002-06-26 EP disclosed
US-6368814-B1 TRICYCLIC ANTIDEPRESSANTS AND METABOLITES THEREOF ROCHE DIAGNOSTICS CORPORATION 2002-04-09 US disclosed
US-4399141-A 5-Alkyl or hydroxyalkyl substituted-10,11-dihydro-5H-dibenzo[a,d]cyclohepten-5,10-imines and anticonvulsant use thereof MERCK & CO., INC. (US) 1983-08-16 US disclosed
US-4333920-A Benzalphthalides and broad spectrum sun screens VAN DYK & COMPANY, INC. (US) 1982-06-08 US disclosed