SCHEMBL4679711

SCHEMBL4679711

CCCN(CC1CCN(C(=O)N2CCOCC2)CC1)[C@H](C)Cc1cccc(NC(=O)c2ccc(OC)cc2)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.46
RAB9A P51151 4/20 0.46
SMN1; SMN2 Q16637 4/20 0.46
LMNA P02545 3/20 0.46
TP53 P04637 3/20 0.46
HIF1A Q16665 1/20 0.43
EPAS1 Q99814 1/20 0.43
ACKR3 P25106 2/20 0.42
ALDH1A1 P00352 3/20 0.41
MAPK1 P28482 1/20 0.41
AURKA O14965 1/20 0.40
RPS6KB1 P23443 1/20 0.40
AURKB Q96GD4 1/20 0.40
KDM4E B2RXH2 1/20 0.40
CASP3 P42574 1/20 0.40
SENP7 Q9BQF6 1/20 0.40
POLB P06746 1/20 0.40
SLC1A3 P43003 1/20 0.40
SLC1A2 P43004 1/20 0.40
SLC1A1 P43005 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4679382 1.00 NPC1 (0.46) NPC1RAB9ASMN1; SMN2LMNATP53
Hydrochloric Acid SCHEMBL4680076 0.95 NPC1 (0.44) NPC1RAB9ASMN1; SMN2LMNATP53
Hydrochloric Acid SCHEMBL4682831 0.94 NPC1 (0.44) NPC1RAB9ASMN1; SMN2LMNATP53
SCHEMBL4677928 0.93 LMNA (0.46) NPC1RAB9ASMN1; SMN2LMNATP53
SCHEMBL4680175 0.93 SMN1; SMN2 (0.42) NPC1RAB9ASMN1; SMN2LMNATP53
Hydrochloric Acid SCHEMBL4679163 0.93 NPC1 (0.47) NPC1RAB9ASMN1; SMN2LMNATP53
SCHEMBL4678644 0.92 CYP2C19 (0.41) NPC1RAB9ASMN1; SMN2LMNATP53
SCHEMBL4682972 0.92 PPARA (0.40) NPC1RAB9ASMN1; SMN2LMNATP53
SCHEMBL4679962 0.91 ACKR3 (0.45) NPC1RAB9ASMN1; SMN2LMNATP53
SCHEMBL4679955 0.91 ACKR3 (0.45) NPC1RAB9ASMN1; SMN2LMNATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1058680-B1 2-ARYLETHYL-(PIPERIDIN-4-YLMETHYL)AMINE DERIVATIVES AS MUSCARINIC RECEPTOR ANTAGONISTS HOFFMANN LA ROCHE (CH) 2008-07-09 EP disclosed
US-6319920-B1 MUSCARINIC RECEPTOR ANTAGONIST USED IN GASTROINTESTINAL, GENITOURINARY TRACT, RESPIRATORY TRACT, CARDIOVASCULAR SYSTEM, CENTRAL NERVOUS SYSTEM DISORDERS AND IN ANESTHESIOLOGY AND OPHTHALMOLOGY SYNTEX (U.S.A.) LLC 2001-11-20 US disclosed