SCHEMBL467989

SCHEMBL467989

CCCCCc1nc2c(C(N)=O)cccc2[nH]1.NC(=O)c1cccc2[nH]c(-c3ccc(O)cc3)nc12

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 18/20 0.71
DHODH Q02127 1/20 0.58
AURKB Q96GD4 2/20 0.58
AURKA O14965 1/20 0.58
PLA2G2A P14555 1/20 0.57
ALOX15 P16050 1/20 0.57
PTGS2 P35354 1/20 0.57
PARP2 Q9UGN5 1/20 0.56
PLK4 O00444 1/20 0.56
MAPK13 O15264 1/20 0.56
DYRK3 O43781 1/20 0.56
ROCK2 O75116 1/20 0.56
RPS6KA5 O75582 1/20 0.56
PRKD3 O94806 1/20 0.56
MAP4K4 O95819 1/20 0.56
CHEK2 O96017 1/20 0.56
PIM1 P11309 1/20 0.56
PHKG2 P15735 1/20 0.56
PRKACA P17612 1/20 0.56
RPS6KB1 P23443 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL461964 0.88 PARP1 (0.58) PARP1PARP2
SCHEMBL423551 0.84 PARP1 (1.00) PARP1DHODHAURKBPLA2G2AALOX15
SCHEMBL29380664 0.84 PARP1 (1.00) PARP1DHODHAURKBPLA2G2AALOX15
SCHEMBL5630156 0.80 PARP1 (0.61) PARP1AURKBAURKAPARP2
SCHEMBL12385320 0.80 PARP1 (0.62) PARP1DHODHAURKBPARP2PLK4
SCHEMBL28263632 0.78 KDM4E (0.50) PARP1DHODH
SCHEMBL29180021 0.76 PARP1 (0.73) PARP1DHODHAURKBAURKAPLA2G2A
SCHEMBL18252746 0.76 PARP1 (0.78) PARP1DHODHAURKBPLA2G2AALOX15
SCHEMBL29180033 0.75 PARP1 (0.68) PARP1DHODHAURKBAURKAPLA2G2A
SCHEMBL30811237 0.75 PARP1 (0.68) PARP1DHODHAURKBAURKAPLA2G2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2387403-A1 METHOD OF TREATING CANCER Academisch Medisch Centrum bij de Universiteit van Amsterdam (NL) 2011-11-23 EP disclosed
US-20110253692-A1 Electrical heater for vehicle windshields and windows SCHAUBLE RICHARD EGON 2011-10-20 US disclosed