SCHEMBL4681635

SCHEMBL4681635

CC(=O)NC1CCN(C[O])CC1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 3/20 0.44
ATM Q13315 1/20 0.41
EPHX2 P34913 3/20 0.41
EPHX1 P07099 2/20 0.41
CHRM1 P11229 3/20 0.40
DRD2 P14416 2/20 0.40
DRD3 P35462 1/20 0.40
ALDH1A1 P00352 2/20 0.40
CA1 P00915 2/20 0.39
CA2 P00918 2/20 0.39
CA12 O43570 1/20 0.39
CA9 Q16790 1/20 0.39
KDM4E B2RXH2 1/20 0.39
CYP2D6 P10635 1/20 0.39
HTR2A P28223 1/20 0.39
MCHR1 Q99705 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4681639 0.88 LTA4H (0.44) LTA4HATMEPHX2EPHX1CHRM1
SCHEMBL20194151 0.86 LTA4H (0.43) LTA4HATMEPHX2EPHX1CHRM1
SCHEMBL12337290 0.84 EPHX1 (0.54) LTA4HATMEPHX2EPHX1ALDH1A1
SCHEMBL14527915 0.82 LTA4H (0.43) LTA4HATMEPHX2EPHX1CHRM1
SCHEMBL4681787 0.82 CHRM1 (0.48) LTA4HATMEPHX2EPHX1CHRM1
SCHEMBL669964 0.81 LTA4H (0.45) LTA4HDRD2DRD3ALDH1A1
SCHEMBL13136091 0.81 EPHX1 (0.56) LTA4HEPHX2EPHX1ALDH1A1KDM4E
SCHEMBL8144691 0.81 LTA4H (0.48) LTA4HEPHX2EPHX1CHRM1DRD2
SCHEMBL29602619 0.79 PIK3CD (0.50) LTA4HATMCHRM1DRD2DRD3
SCHEMBL7284403 0.79 LTA4H (0.41) LTA4HATMEPHX2EPHX1CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1902717-A2 Vasopressin antagonist and oxytocin antagonist Otsuka Pharmaceutical Company, Limited (JP) 2008-03-26 EP disclosed
EP-0620003-B1 VASOPRESSIN ANTAGONIST AND OXYTOCIN ANTAGONIST OTSUKA PHARMA CO LTD (JP) 2008-01-16 EP disclosed
US-5753644-A Vasopressin antagonist and oxytocin antagonist OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1998-05-19 US disclosed
US-5622947-A VASODILATORS, HYPOTENSIVE AGENTS, DIURETICS, PLATELET AGGLUTINATION INHIBITORS; ALSO USED TO PREVENT PREMATURE BIRTH, TREAT DYSMENORRHEA OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1997-04-22 US disclosed
EP-0620003-A1 VASOPRESSIN ANTAGONIST AND OXYTOCIN ANTAGONIST OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-10-19 EP disclosed