SCHEMBL4682633

SCHEMBL4682633

CCCN(CC1CCN(S(C)(=O)=O)CC1)[C@@H](C)Cc1cccc(NC(=O)c2ccc(F)cc2)c1

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ACKR3 P25106 9/20 0.47
CYP2D6 P10635 1/20 0.45
HTR1F P30939 1/20 0.41
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
ALDH1A1 P00352 3/20 0.41
MAPT P10636 2/20 0.39
RECQL P46063 1/20 0.39
MAPK1 P28482 1/20 0.39
HTT P42858 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
PPARA Q07869 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4682634 1.00 ACKR3 (0.47) ACKR3CYP2D6HTR1FMEN1KMT2A
Hydrochloric Acid SCHEMBL4685659 0.92 TRPV4 (0.46) ACKR3CYP2D6MAPTSMN1; SMN2
Hydrochloric Acid SCHEMBL4685656 0.92 TRPV4 (0.46) ACKR3CYP2D6MAPTSMN1; SMN2
Hydrochloric Acid SCHEMBL4681798 0.91 ACKR3 (0.47) ACKR3CYP2D6MEN1KMT2AALDH1A1
Hydrochloric Acid SCHEMBL4681803 0.91 ACKR3 (0.47) ACKR3CYP2D6MEN1KMT2AALDH1A1
Hydrochloric Acid SCHEMBL4679511 0.91 CYP2D6 (0.44) ACKR3CYP2D6MEN1KMT2AALDH1A1
Hydrochloric Acid SCHEMBL4679507 0.91 CYP2D6 (0.44) ACKR3CYP2D6MEN1KMT2AALDH1A1
Hydrochloric Acid SCHEMBL4683274 0.89 ACKR3 (0.43) ACKR3CYP2D6ALDH1A1
Hydrochloric Acid SCHEMBL4683276 0.89 ACKR3 (0.43) ACKR3CYP2D6ALDH1A1
Trifluoroacetic Acid SCHEMBL4683847 0.89 NR1H4 (0.43) ACKR3CYP2D6MEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1058680-B1 2-ARYLETHYL-(PIPERIDIN-4-YLMETHYL)AMINE DERIVATIVES AS MUSCARINIC RECEPTOR ANTAGONISTS HOFFMANN LA ROCHE (CH) 2008-07-09 EP disclosed
US-6319920-B1 MUSCARINIC RECEPTOR ANTAGONIST USED IN GASTROINTESTINAL, GENITOURINARY TRACT, RESPIRATORY TRACT, CARDIOVASCULAR SYSTEM, CENTRAL NERVOUS SYSTEM DISORDERS AND IN ANESTHESIOLOGY AND OPHTHALMOLOGY SYNTEX (U.S.A.) LLC 2001-11-20 US disclosed