SCHEMBL4682895

SCHEMBL4682895

OCCCCCCSc1ccncn1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.42
HTT P42858 1/20 0.42
GFER P55789 1/20 0.42
KMT2A Q03164 1/20 0.42
MAPK14 Q16539 3/20 0.37
CA2 P00918 3/20 0.37
GSTP1 P09211 3/20 0.36
GSTM2 P28161 3/20 0.36
HSP90AA1 P07900 1/20 0.35
ALDH1A1 P00352 2/20 0.33
GPR84 Q9NQS5 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
PLA2G7 Q13093 1/20 0.32
P2RX7 Q99572 1/20 0.32
KDM4E B2RXH2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4687649 0.98 HTT (0.43) PKMHTTGFERKMT2AMAPK14
SCHEMBL7350714 0.93 HTT (0.44) PKMHTTGFERKMT2AMAPK14
SCHEMBL7354366 0.87 KMT2A (0.47) PKMHTTGFERKMT2AMAPK14
SCHEMBL4682892 0.83 HTT (0.42) PKMHTTGFERKMT2AHSP90AA1
SCHEMBL4687648 0.81 KMT2A (0.43) PKMHTTGFERKMT2AHSP90AA1
SCHEMBL8906020 0.79 HTT (0.41) PKMHTTGFERKMT2AHSP90AA1
SCHEMBL7350710 0.79 HTT (0.44) PKMHTTGFERKMT2AHSP90AA1
SCHEMBL4685852 0.77 ALDH1A1 (0.56) PKMKMT2AALDH1A1L3MBTL1KDM4E
SCHEMBL4684788 0.77 ALDH1A1 (0.56) PKMKMT2AALDH1A1L3MBTL1KDM4E
SCHEMBL4687627 0.75 ALDH1A1 (0.57) PKMKMT2AALDH1A1L3MBTL1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1902717-A2 Vasopressin antagonist and oxytocin antagonist Otsuka Pharmaceutical Company, Limited (JP) 2008-03-26 EP disclosed
EP-0620003-B1 VASOPRESSIN ANTAGONIST AND OXYTOCIN ANTAGONIST OTSUKA PHARMA CO LTD (JP) 2008-01-16 EP disclosed
US-5753644-A Vasopressin antagonist and oxytocin antagonist OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1998-05-19 US disclosed
US-5622947-A VASODILATORS, HYPOTENSIVE AGENTS, DIURETICS, PLATELET AGGLUTINATION INHIBITORS; ALSO USED TO PREVENT PREMATURE BIRTH, TREAT DYSMENORRHEA OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1997-04-22 US disclosed
EP-0620003-A1 VASOPRESSIN ANTAGONIST AND OXYTOCIN ANTAGONIST OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-10-19 EP disclosed