SCHEMBL4683608

SCHEMBL4683608

CCC(C)C(NC(=O)N(C)Cc1ccccn1)C(=O)OC

nearest known ligand 0.55

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CA2 P00918 2/20 0.55
POLB P06746 3/20 0.46
ALDH1A1 P00352 6/20 0.45
HTT P42858 1/20 0.44
NOS3 P29474 3/20 0.43
NOS1 P29475 3/20 0.43
NOS2 P35228 3/20 0.43
MAPT P10636 1/20 0.42
LMNA P02545 1/20 0.41
HDAC6 Q9UBN7 4/20 0.40
HDAC1 Q13547 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4683611 1.00 CA2 (0.55) CA2POLBALDH1A1HTTNOS3
SCHEMBL4676249 0.91 CA2 (0.62) CA2POLBALDH1A1LMNAHDAC6
SCHEMBL4676251 0.91 CA2 (0.62) CA2POLBALDH1A1LMNAHDAC6
SCHEMBL27395775 0.88 CA2 (0.60) CA2POLBALDH1A1MAPT
SCHEMBL7302427 0.88 CA2 (0.60) CA2POLBALDH1A1MAPT
SCHEMBL7393135 0.88 CA2 (0.60) CA2POLBALDH1A1MAPT
SCHEMBL8660662 0.84 CA2 (0.60) CA2POLBALDH1A1LMNA
SCHEMBL4679457 0.83 CA2 (0.46) CA2POLBALDH1A1HTTMAPT
SCHEMBL4679453 0.83 CA2 (0.46) CA2POLBALDH1A1HTTMAPT
SCHEMBL4683895 0.81 CA2 (0.67) CA2POLBALDH1A1MAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0997459-B1 Intermediates for preparing retroviral protease inhibiting compounds ABBOTT LAB (US) 2008-11-26 EP disclosed
EP-0486948-B1 Retroviral protease inhibiting compounds ABBOTT LAB (US) 2000-10-04 EP disclosed
US-5648497-A Retroviral protease inhibiting compounds ABBOTT LABORAOTRIES (US) 1997-07-15 US disclosed
US-5616714-A PYRIDYL, THIAZOLYL-SUBSTITUTED AMINO ACID DERIVATIVES ABBOTT LABORATORIES (US) 1997-04-01 US disclosed
US-5597926-A Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1997-01-28 US disclosed
US-5554783-A (2R, 3R, 4S, 5S)-3-ACETOXY-2,5-BIS/BENZYLOXYCARBONYLAMINO/ -4-BROMO-1,5-DIPHENYLHEXANE ABBOTT LABORATORIES (US) 1996-09-10 US disclosed
US-5541334-A TREATING HIV ABBOTT LABORATORIES (US) 1996-07-30 US disclosed
US-5354866-A Treating HIV infections ABBOTT LABORATORIES (US) 1994-10-11 US disclosed
EP-0486948-A2 Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1992-05-27 EP disclosed