SCHEMBL4684100

SCHEMBL4684100

OCCCCc1nn[nH]n1

nearest known ligand 0.75

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 2/20 0.75
ALDH1A1 P00352 1/20 0.71
LMNA P02545 1/20 0.71
CTH P32929 1/20 0.49
TBXAS1 P24557 5/20 0.46
EPHX2 P34913 2/20 0.42
GRIN2D O15399 1/20 0.42
GRIN3B O60391 1/20 0.42
GRIN1 Q05586 1/20 0.42
GRIN2A Q12879 1/20 0.42
GRIN2B Q13224 1/20 0.42
GRIN2C Q14957 1/20 0.42
GRIN3A Q8TCU5 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
NAALAD2 Q9Y3Q0 1/20 0.41
KDM6B O15054 1/20 0.40
KDM4A O75164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4682596 0.98 L3MBTL1 (0.79) L3MBTL1ALDH1A1LMNACTHTBXAS1
SCHEMBL2948127 0.84
SCHEMBL9986002 0.78 L3MBTL1 (0.79) L3MBTL1ALDH1A1LMNACTHTBXAS1
SCHEMBL14518629 0.77 L3MBTL1 (0.79) L3MBTL1ALDH1A1LMNACTHTBXAS1
SCHEMBL20936411 0.77 L3MBTL1 (0.79) L3MBTL1ALDH1A1LMNACTHTBXAS1
SCHEMBL6000049 0.77 L3MBTL1 (0.79) L3MBTL1ALDH1A1LMNACTHTBXAS1
SCHEMBL4682373 0.76
SCHEMBL30843332 0.75 L3MBTL1 (0.68) L3MBTL1ALDH1A1LMNACTHTBXAS1
SCHEMBL13780257 0.75 L3MBTL1 (0.62) L3MBTL1ALDH1A1LMNACTHTBXAS1
SCHEMBL16522419 0.74 L3MBTL1 (0.67) L3MBTL1ALDH1A1LMNACTHTBXAS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1902717-A2 Vasopressin antagonist and oxytocin antagonist Otsuka Pharmaceutical Company, Limited (JP) 2008-03-26 EP disclosed
EP-0620003-B1 VASOPRESSIN ANTAGONIST AND OXYTOCIN ANTAGONIST OTSUKA PHARMA CO LTD (JP) 2008-01-16 EP disclosed
US-5753644-A Vasopressin antagonist and oxytocin antagonist OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1998-05-19 US disclosed
US-5622947-A VASODILATORS, HYPOTENSIVE AGENTS, DIURETICS, PLATELET AGGLUTINATION INHIBITORS; ALSO USED TO PREVENT PREMATURE BIRTH, TREAT DYSMENORRHEA OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1997-04-22 US disclosed
EP-0620003-A1 VASOPRESSIN ANTAGONIST AND OXYTOCIN ANTAGONIST OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-10-19 EP disclosed