SCHEMBL4685609

SCHEMBL4685609

CCCN(CC1CCN(S(C)(=O)=O)CC1)C(C)Cc1cccc(NS(=O)(=O)N(C)C)c1

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.49
PARP1 P09874 1/20 0.35
ALDH1A1 P00352 2/20 0.35
POLB P06746 1/20 0.34
ACP1 P24666 1/20 0.34
MEN1 O00255 3/20 0.34
KMT2A Q03164 3/20 0.34
RORC P51449 2/20 0.34
HTT P42858 1/20 0.34
PDE4A P27815 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
MCHR1 Q99705 2/20 0.33
FABP6 P51161 1/20 0.33
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8132866 0.92 CYP2D6 (0.51) CYP2D6ALDH1A1ACP1RORCL3MBTL1
Hydrochloric Acid SCHEMBL4679793 0.91 CYP2D6 (0.51) CYP2D6ALDH1A1ACP1RORCL3MBTL1
SCHEMBL4683282 0.86 CYP2D6 (0.47) CYP2D6ALDH1A1MEN1KMT2AHTT
SCHEMBL4678497 0.85 CYP2D6 (0.51) CYP2D6ALDH1A1POLBMEN1KMT2A
Hydrochloric Acid SCHEMBL4682628 0.84 CYP2D6 (0.48) CYP2D6ALDH1A1POLBMEN1KMT2A
Hydrochloric Acid SCHEMBL4682834 0.84 CYP2D6 (0.48) CYP2D6PARP1ALDH1A1POLBMEN1
SCHEMBL4685281 0.83 CYP2D6 (0.54) CYP2D6ALDH1A1POLBMEN1KMT2A
SCHEMBL4685621 0.83 CYP2D6 (0.47) CYP2D6ALDH1A1POLBMEN1KMT2A
SCHEMBL4679978 0.81 ACKR3 (0.46) CYP2D6ALDH1A1POLBMEN1KMT2A
SCHEMBL4682819 0.81 CYP2D6 (0.47) CYP2D6ALDH1A1POLBMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1058680-B1 2-ARYLETHYL-(PIPERIDIN-4-YLMETHYL)AMINE DERIVATIVES AS MUSCARINIC RECEPTOR ANTAGONISTS HOFFMANN LA ROCHE (CH) 2008-07-09 EP disclosed
US-6319920-B1 MUSCARINIC RECEPTOR ANTAGONIST USED IN GASTROINTESTINAL, GENITOURINARY TRACT, RESPIRATORY TRACT, CARDIOVASCULAR SYSTEM, CENTRAL NERVOUS SYSTEM DISORDERS AND IN ANESTHESIOLOGY AND OPHTHALMOLOGY SYNTEX (U.S.A.) LLC 2001-11-20 US disclosed