SCHEMBL4685809

SCHEMBL4685809

CC(C[O])CSc1ccccn1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.53
HPGD P15428 3/20 0.53
MEN1 O00255 2/20 0.53
TSHR P16473 1/20 0.53
ALDH1A1 P00352 6/20 0.47
RAB9A P51151 6/20 0.47
NPC1 O15118 5/20 0.47
TDP1 Q9NUW8 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
LMNA P02545 1/20 0.46
SMN1; SMN2 Q16637 2/20 0.45
HSD17B10 Q99714 2/20 0.45
KDM4E B2RXH2 1/20 0.45
ALOX15 P16050 1/20 0.45
EHMT2 Q96KQ7 1/20 0.45
EHMT1 Q9H9B1 1/20 0.45
APOBEC3G Q9HC16 1/20 0.45
MAPT P10636 1/20 0.44
PKM P14618 1/20 0.44
POLB P06746 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4685810 0.82 KMT2A (0.56) KMT2AHPGDMEN1TSHRALDH1A1
SCHEMBL2608954 0.81 KMT2A (0.58) KMT2AHPGDMEN1TSHRALDH1A1
SCHEMBL7287371 0.79 GAA (0.40) KMT2AHPGDTSHRALDH1A1RAB9A
Ammonia Solution, Strong SCHEMBL7245354 0.79 KMT2A (0.57) KMT2AHPGDMEN1TSHRALDH1A1
SCHEMBL8427849 0.79 KMT2A (0.57) KMT2AHPGDMEN1TSHRALDH1A1
SCHEMBL4681376 0.79 KMT2A (0.41) KMT2AHPGDMEN1TSHRALDH1A1
SCHEMBL4687320 0.77
SCHEMBL7421414 0.76 KMT2A (0.57) KMT2AHPGDMEN1TSHRALDH1A1
SCHEMBL19787804 0.76 HPGD (0.57) KMT2AHPGDMEN1TSHRALDH1A1
Acetic Acid SCHEMBL28119023 0.76 ALDH1A1 (0.57) KMT2AHPGDMEN1TSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1902717-A2 Vasopressin antagonist and oxytocin antagonist Otsuka Pharmaceutical Company, Limited (JP) 2008-03-26 EP disclosed
EP-0620003-B1 VASOPRESSIN ANTAGONIST AND OXYTOCIN ANTAGONIST OTSUKA PHARMA CO LTD (JP) 2008-01-16 EP disclosed
US-5753644-A Vasopressin antagonist and oxytocin antagonist OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1998-05-19 US disclosed
US-5622947-A VASODILATORS, HYPOTENSIVE AGENTS, DIURETICS, PLATELET AGGLUTINATION INHIBITORS; ALSO USED TO PREVENT PREMATURE BIRTH, TREAT DYSMENORRHEA OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1997-04-22 US disclosed
EP-0620003-A1 VASOPRESSIN ANTAGONIST AND OXYTOCIN ANTAGONIST OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-10-19 EP disclosed