SCHEMBL4685869

SCHEMBL4685869

[CH2]C(C)CC1CCN(C)C1

nearest known ligand 0.41

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
NCF1 P14598 1/20 0.41
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33
CHRM2 P08172 1/20 0.30
CHRM1 P11229 1/20 0.30
CHRM3 P20309 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9036617 0.88 CHRM2 (0.36) NCF1CYP2D6CHRM2CHRM1CHRM3
SCHEMBL8235125 0.82 NCF1 (0.44) NCF1CYP1A2CYP2D6CHRM2CHRM1
SCHEMBL23645702 0.82 NCF1 (0.44) NCF1CYP1A2CYP2D6CHRM2CHRM1
SCHEMBL22020557 0.82 NCF1 (0.44) NCF1CYP1A2CYP2D6CHRM2CHRM1
SCHEMBL30831689 0.80 NCF1 (0.48) NCF1CYP1A2CYP2D6CHRM2CHRM1
SCHEMBL24428727 0.78 NCF1 (0.41) NCF1CYP1A2CYP2D6CHRM2CHRM1
SCHEMBL23473264 0.78 NCF1 (0.38) NCF1CYP1A2CYP2D6
SCHEMBL14546268 0.77 NCF1 (0.40) NCF1CYP1A2CYP2D6
SCHEMBL27267519 0.75 NCF1 (0.39) NCF1CYP1A2CYP2D6
SCHEMBL95411 0.73

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1902717-A2 Vasopressin antagonist and oxytocin antagonist Otsuka Pharmaceutical Company, Limited (JP) 2008-03-26 EP disclosed
EP-0620003-B1 VASOPRESSIN ANTAGONIST AND OXYTOCIN ANTAGONIST OTSUKA PHARMA CO LTD (JP) 2008-01-16 EP disclosed
CN-1306935-C Vasopressin antagonist and oxytocin antagonist OTASUKA PHARMACEUTICAL CO LTD (JP) 2007-03-28 CN disclosed
CN-1039999-C Vasopressin antagonist and oxytocin antagonist, process for their preparation and pharmaceutical compositions containing them OTSUKA CHEMICAL CO LTD (JP) 1998-09-30 CN disclosed
CN-1183277-A Vasopressin antagonist and oxytocin antagonist OTASUKA PHARMACEUTICAL CO LTD (JP) 1998-06-03 CN disclosed
US-5753644-A Vasopressin antagonist and oxytocin antagonist OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1998-05-19 US disclosed
US-5622947-A VASODILATORS, HYPOTENSIVE AGENTS, DIURETICS, PLATELET AGGLUTINATION INHIBITORS; ALSO USED TO PREVENT PREMATURE BIRTH, TREAT DYSMENORRHEA OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1997-04-22 US disclosed
CN-1098716-A Vasopressin antagonists and oxytocin antagonists OTSUKA CHEMICAL CO LTD (JP) 1995-02-15 CN disclosed
EP-0620003-A1 VASOPRESSIN ANTAGONIST AND OXYTOCIN ANTAGONIST OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-10-19 EP disclosed