SCHEMBL4686337

SCHEMBL4686337

COc1cc(NC(=O)c2ccccc2Cl)ccc1C(=O)N1c2ccc(Cl)cc2C(CCN(C)CCO)CCC1CC(N)=O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM4 Q14833 8/20 0.38
ALDH1A1 P00352 3/20 0.38
KDM4E B2RXH2 3/20 0.38
KMT2A Q03164 2/20 0.38
MAPT P10636 4/20 0.37
SPTLC2 O15270 1/20 0.37
SMN1; SMN2 Q16637 3/20 0.36
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
MEN1 O00255 1/20 0.36
POLB P06746 1/20 0.36
AVPR2 P30518 3/20 0.36
PTGS2 P35354 1/20 0.36
CHRM1 P11229 2/20 0.36
CHRM5 P08912 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4688309 0.87 AVPR2 (0.41) GRM4ALDH1A1KDM4EKMT2AMAPT
SCHEMBL4686328 0.77 AVPR2 (0.48) GRM4SPTLC2AVPR2CHRM1AVPR1A
SCHEMBL7334873 0.77 AVPR2 (0.54) GRM4ALDH1A1KDM4EKMT2ASPTLC2
SCHEMBL4743938 0.76 AVPR2 (0.50) GRM4SPTLC2AVPR2CHRM1AVPR1A
SCHEMBL4743947 0.75 GRM4 (0.39) GRM4ALDH1A1KDM4EKMT2AMAPT
SCHEMBL7354159 0.75 AVPR2 (0.57) GRM4SPTLC2AVPR2CHRM1CHRM5
SCHEMBL7334875 0.75 GRM4 (0.45) GRM4ALDH1A1KDM4EKMT2AMAPT
SCHEMBL4695541 0.73 AVPR2 (0.53) GRM4ALDH1A1KDM4EKMT2ASPTLC2
SCHEMBL4743943 0.72 AVPR2 (0.49) GRM4SPTLC2AVPR2CHRM1AVPR1A
SCHEMBL4681402 0.72 AVPR2 (0.55) GRM4SPTLC2AVPR2CHRM1AVPR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1902717-A2 Vasopressin antagonist and oxytocin antagonist Otsuka Pharmaceutical Company, Limited (JP) 2008-03-26 EP disclosed
EP-0620003-B1 VASOPRESSIN ANTAGONIST AND OXYTOCIN ANTAGONIST OTSUKA PHARMA CO LTD (JP) 2008-01-16 EP disclosed
US-5622947-A VASODILATORS, HYPOTENSIVE AGENTS, DIURETICS, PLATELET AGGLUTINATION INHIBITORS; ALSO USED TO PREVENT PREMATURE BIRTH, TREAT DYSMENORRHEA OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1997-04-22 US disclosed