SCHEMBL4687017

SCHEMBL4687017

C/C(=C\C(=O)O)Nc1cccc(C)c1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 3/20 0.64
KMT2A Q03164 5/20 0.54
MEN1 O00255 4/20 0.54
RXFP1 Q9HBX9 1/20 0.54
MAOB P27338 3/20 0.54
MAOA P21397 2/20 0.54
EGFR P00533 1/20 0.54
MMP1 P03956 1/20 0.54
MMP2 P08253 1/20 0.54
MMP9 P14780 1/20 0.54
SMN1; SMN2 Q16637 3/20 0.54
NPC1 O15118 2/20 0.54
TP53 P04637 2/20 0.54
MAPT P10636 2/20 0.54
RAB9A P51151 2/20 0.54
HTT P42858 1/20 0.54
NPSR1 Q6W5P4 1/20 0.54
ALDH1A1 P00352 1/20 0.53
MAPK1 P28482 2/20 0.52
KCNK3 O14649 2/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4687023 1.00 HSD17B10 (0.64) HSD17B10KMT2AMEN1RXFP1MAOB
SCHEMBL4687025 1.00 HSD17B10 (0.64) HSD17B10KMT2AMEN1RXFP1MAOB
SCHEMBL5477342 0.88 HSD17B10 (0.66) HSD17B10KMT2AMEN1RXFP1MAOB
SCHEMBL5477339 0.88 HSD17B10 (0.66) HSD17B10KMT2AMEN1RXFP1MAOB
SCHEMBL14520811 0.88 HSD17B10 (0.66) HSD17B10KMT2AMEN1RXFP1MAOB
SCHEMBL14482921 0.82 MAPT (0.63) HSD17B10KMT2AMEN1SMN1; SMN2NPC1
SCHEMBL1975201 0.82 MAPT (0.63) HSD17B10KMT2AMEN1SMN1; SMN2NPC1
SCHEMBL1975200 0.82 MAPT (0.63) HSD17B10KMT2AMEN1SMN1; SMN2NPC1
SCHEMBL29217657 0.82 MEN1 (0.56) HSD17B10KMT2AMEN1MMP1MMP2
SCHEMBL29217646 0.82 MAPT (0.59) HSD17B10KMT2AMEN1MAOBMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1537081-B1 DIHYDROPYRIDINE DERIVATIVES FOR USE AS HUMAN NEUTROPHIL ELASTASE INHIBITORS BAYER HEALTHCARE AG (DE) 2008-10-15 EP disclosed
EP-1458682-B1 1,4-DIHYDRO-1,4-DIPHENYLPYRIDINE DERIVATIVES BAYER HEALTHCARE AG (DE) 2006-08-30 EP disclosed
EP-1537081-A1 DIHYDROPYRIDINE DERIVATIVES FOR USE AS HUMAN NEUTROPHIL ELASTASE INHIBITORS Bayer HealthCare AG (DE) 2005-06-08 EP disclosed
EP-1458682-A1 1,4-DIHYDRO-1,4-DIPHENYLPYRIDINE DERIVATIVES Bayer HealthCare AG (DE) 2004-09-22 EP disclosed
WO-2004020412-A1 DIHYDROPYRIDINE DERIVATIVES FOR USE AS HUMAN NEUTROPHIL ELASTASE INHIBITORS BAYER HEALTHCARE AG (DE) 2004-03-11 WO disclosed
WO-2003053930-A1 1,4-DIHYDRO-1,4-DIPHENYLPYRIDINE DERIVATIVES BAYER HEALTHCARE AG (DE) 2003-07-03 WO disclosed