SCHEMBL4687699

SCHEMBL4687699

CCCCCNCc1ccc(Oc2cnc(OC(N)=O)cn2)c(OC)c1

nearest known ligand 0.62

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.54
HDAC3 O15379 1/20 0.52
HDAC1 Q13547 1/20 0.52
HDAC2 Q92769 1/20 0.52
HDAC8 Q9BY41 1/20 0.52
S1PR2 O95136 1/20 0.52
S1PR1 P21453 1/20 0.52
S1PR3 Q99500 1/20 0.52
LPAR2 Q9HBW0 1/20 0.52
POLB P06746 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.49
EPHX2 P34913 1/20 0.48
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
HTT P42858 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3693840 0.90 KDM4E (0.52) KDM4EHDAC3HDAC1HDAC2HDAC8
SCHEMBL3692313 0.86 OPRM1 (0.53) KDM4EHDAC3HDAC1HDAC2HDAC8
SCHEMBL13773093 0.85 S1PR2 (0.54) KDM4EHDAC3HDAC1HDAC2HDAC8
SCHEMBL3692559 0.85 S1PR2 (0.54) KDM4EHDAC3HDAC1HDAC2HDAC8
SCHEMBL3689803 0.84 OPRM1 (0.51) KDM4EHDAC3HDAC1HDAC2HDAC8
SCHEMBL3694884 0.83 OPRM1 (0.54) KDM4EHDAC3HDAC1HDAC2HDAC8
SCHEMBL3694672 0.83 S1PR2 (0.52) KDM4EHDAC3HDAC1HDAC2HDAC8
SCHEMBL3697283 0.83 S1PR2 (0.52) KDM4EHDAC3HDAC1HDAC2HDAC8
SCHEMBL3693831 0.82 KDM4E (0.50) KDM4EHDAC3HDAC1HDAC2HDAC8
SCHEMBL12018423 0.82 KDM4E (0.52) KDM4EHDAC3HDAC1HDAC2HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1562595-B1 DIARYL ETHERS AS OPIOID RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-05-21 EP disclosed