SCHEMBL4687741

SCHEMBL4687741

CCC(CC)NC(=O)Nc1ccc(Oc2ccc(NC(=O)O)cc2COC)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.56
TAS1R3 Q7RTX0 1/20 0.46
TAS1R1 Q7RTX1 1/20 0.46
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
MAPK1 P28482 1/20 0.41
ALDH1A1 P00352 2/20 0.40
MEN1 O00255 3/20 0.39
MAPT P10636 3/20 0.39
KMT2A Q03164 3/20 0.39
GAA P10253 2/20 0.39
LMNA P02545 1/20 0.38
TP53 P04637 1/20 0.38
HTT P42858 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
HIF1A Q16665 1/20 0.38
MTNR1B P49286 1/20 0.38
NPY5R Q15761 1/20 0.38
FPR2 P25090 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4236335 0.89 PKM (0.53) PKMTAS1R3TAS1R1CYP2C9CYP2C19
SCHEMBL4234125 0.87 PKM (0.56) PKMTAS1R3TAS1R1CYP2C9CYP2C19
SCHEMBL4242559 0.86 PKM (0.49) PKMTAS1R3TAS1R1MAPK1MEN1
SCHEMBL4683708 0.86 PKM (0.63) PKMTAS1R3TAS1R1CYP2C9CYP2C19
SCHEMBL5149842 0.86 PKM (0.63) PKMTAS1R3TAS1R1CYP2C9CYP2C19
SCHEMBL4236717 0.85 PKM (0.54) PKMTAS1R3TAS1R1CYP2C9CYP2C19
SCHEMBL4685639 0.83 MAPT (0.40) MAPK1ALDH1A1MEN1MAPTKMT2A
SCHEMBL4238927 0.82 PKM (0.54) PKMTAS1R3TAS1R1CYP2C9CYP2C19
SCHEMBL4687749 0.81 EPHX1 (0.49) PKMALDH1A1MAPTKMT2ALMNA
SCHEMBL4242160 0.81 PKM (0.46) PKMTAS1R3TAS1R1ALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1879887-A2 NPY ANTAGONISTS, PREPARATION AND USE Cerep (FR) 2008-01-23 EP disclosed
WO-2007071840-A2 COMPOUNDS BASED ON FOUR AROMATIC RINGS, PREPARATION AND USES THEREOF CEREP (FR) 2007-06-28 WO disclosed
WO-2006108965-A2 NPY ANTAGONISTS, PREPARATION AND USE CEREP (FR) 2006-10-19 WO disclosed