SCHEMBL4688028

SCHEMBL4688028

FC(F)(F)c1ccccc1CN1CCC(NC2CCOCC2)C1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 8/20 0.47
ALDH1A1 P00352 7/20 0.47
ATM Q13315 2/20 0.47
SIGMAR1 Q99720 1/20 0.47
KMT2A Q03164 1/20 0.45
MAPT P10636 1/20 0.44
POLB P06746 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
TACR1 P25103 2/20 0.43
NPSR1 Q6W5P4 2/20 0.43
BCHE P06276 1/20 0.41
ACHE P22303 1/20 0.41
BACE1 P56817 1/20 0.41
TDP1 Q9NUW8 2/20 0.41
RECQL P46063 1/20 0.41
GAA P10253 1/20 0.41
PKM P14618 1/20 0.41
CYP2D6 P10635 1/20 0.41
SLC6A2 P23975 1/20 0.41
SLC6A4 P31645 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3166277 0.81 KDM4E (0.52) KDM4EALDH1A1ATMSIGMAR1KMT2A
SCHEMBL16269143 0.76 CYP2D6 (0.49) KDM4EALDH1A1ATMSIGMAR1KMT2A
SCHEMBL15859936 0.76 KDM4E (0.67) KDM4EALDH1A1ATMKMT2APOLB
SCHEMBL4488404 0.74 KDM4E (0.56) KDM4EALDH1A1ATMSIGMAR1KMT2A
SCHEMBL29716462 0.72 KDM4E (0.53) KDM4EALDH1A1ATMSIGMAR1KMT2A
SCHEMBL15859935 0.72 KDM4E (0.55) KDM4EALDH1A1ATMKMT2AMAPT
SCHEMBL21101334 0.71 ALDH1A1 (0.56) KDM4EALDH1A1ATMSIGMAR1KMT2A
SCHEMBL15859937 0.71 KDM4E (0.63) KDM4EALDH1A1ATMSIGMAR1KMT2A
SCHEMBL6944191 0.71 KDM4E (0.63) KDM4EALDH1A1ATMSIGMAR1KMT2A
SCHEMBL24529820 0.71 DRD4 (0.53) SIGMAR1POLBPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1638934-B1 3-AMINOPYRROLIDINES AS INHIBITORS OF MONOAMINE UPTAKE LILLY CO ELI (US) 2008-01-09 EP disclosed