SCHEMBL4688358

SCHEMBL4688358

O=C(CCC1CCC[N]1)N1CCCC1

nearest known ligand 0.56

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ATM Q13315 2/20 0.47
ALDH1A1 P00352 3/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
TP53 P04637 1/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
HSD11B1 P28845 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
NPC1 O15118 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8628661 0.85 ATM (0.52) ATMALDH1A1SMN1; SMN2TP53L3MBTL1
SCHEMBL945435 0.76 ATM (0.44) ATMALDH1A1SMN1; SMN2L3MBTL1MEN1
SCHEMBL8484583 0.76 KMT2A (0.42) ALDH1A1TP53MEN1KMT2A
SCHEMBL8483277 0.76 KMT2A (0.45) ATMALDH1A1TP53L3MBTL1MEN1
SCHEMBL8481052 0.74 KMT2A (0.43) ATMALDH1A1TP53L3MBTL1MEN1
SCHEMBL8486542 0.74 KMT2A (0.38) ATMALDH1A1TP53MEN1KMT2A
SCHEMBL2644261 0.74 KMT2A (0.33) L3MBTL1KMT2A
SCHEMBL31487813 0.74 TP53 (0.62) ATMALDH1A1SMN1; SMN2TP53L3MBTL1
SCHEMBL7217209 0.72 TP53 (0.71) ATMALDH1A1SMN1; SMN2TP53MEN1
SCHEMBL3632776 0.71 ALDH1A1 (0.36) ALDH1A1L3MBTL1MEN1KMT2ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1902717-A2 Vasopressin antagonist and oxytocin antagonist Otsuka Pharmaceutical Company, Limited (JP) 2008-03-26 EP disclosed
EP-0620003-B1 VASOPRESSIN ANTAGONIST AND OXYTOCIN ANTAGONIST OTSUKA PHARMA CO LTD (JP) 2008-01-16 EP disclosed
US-5753644-A Vasopressin antagonist and oxytocin antagonist OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1998-05-19 US disclosed
US-5622947-A VASODILATORS, HYPOTENSIVE AGENTS, DIURETICS, PLATELET AGGLUTINATION INHIBITORS; ALSO USED TO PREVENT PREMATURE BIRTH, TREAT DYSMENORRHEA OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1997-04-22 US disclosed
EP-0620003-A1 VASOPRESSIN ANTAGONIST AND OXYTOCIN ANTAGONIST OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-10-19 EP disclosed