SCHEMBL4688487

SCHEMBL4688487

CC(c1ccc(F)cc1)C(CNC(=O)C(C)(C)Oc1cc(C(F)(F)F)ncn1)c1cncc(Br)c1

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 10/20 0.39
AR P10275 1/20 0.31
P2RX7 Q99572 4/20 0.31
TRPA1 O75762 1/20 0.31
CNR2 P34972 1/20 0.31
EGFR P00533 1/20 0.30
DGAT2 Q96PD7 1/20 0.30
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30
EPHX2 P34913 1/20 0.30
CYP2J2 P51589 1/20 0.30
LMNA P02545 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4691568 0.93 CNR1 (0.43) CNR1CNR2CYP2C9
SCHEMBL4692012 0.91 CNR1 (0.41) CNR1P2RX7TRPA1CNR2EPHX2
SCHEMBL4691595 0.87 CNR1 (0.39) CNR1CNR2CYP2C9
SCHEMBL4788252 0.86 CNR1 (0.49) CNR1CNR2DGAT2CYP2C9CYP2C19
SCHEMBL4688592 0.85 CNR1 (0.40) CNR1CNR2CYP2C9
SCHEMBL3374144 0.83 CNR1 (0.57) CNR1CNR2CYP2C9
SCHEMBL4691419 0.82 CNR1 (0.51) CNR1ARCNR2CYP2C9
SCHEMBL4688115 0.81 CNR1 (0.48) CNR1CNR2CYP2C9
SCHEMBL4693237 0.81 CNR1 (0.48) CNR1CNR2CYP2C9
SCHEMBL4694454 0.80 CNR1 (0.47) CNR1CNR2DGAT2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1496838-A4 SUBSTITUTED AMIDES MERCK & CO INC (US) 2008-07-02 EP claimed
EP-1496838-A2 SUBSTITUTED AMIDES Merck & Co., Inc. (US) 2005-01-19 EP claimed
WO-2003077847-A2 SUBSTITUTED AMIDES MERCK & CO., INC. (US) 2003-09-25 WO claimed
EP-1496838-A4 SUBSTITUTED AMIDES MERCK & CO INC (US) 2008-07-02 EP disclosed
EP-1496838-A2 SUBSTITUTED AMIDES Merck & Co., Inc. (US) 2005-01-19 EP disclosed
WO-2003077847-A2 SUBSTITUTED AMIDES MERCK & CO., INC. (US) 2003-09-25 WO disclosed