SCHEMBL4690218

SCHEMBL4690218

CC(Oc1ccc(S(C)(=O)=O)cn1)C(N)=O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.48
KCNH2 Q12809 1/20 0.40
CHRNA7 P36544 1/20 0.40
GPR119 Q8TDV5 1/20 0.38
NNMT P40261 2/20 0.36
ALOX5AP P20292 1/20 0.36
FEN1 P39748 1/20 0.36
LRRK2 Q5S007 1/20 0.36
KDM4E B2RXH2 1/20 0.35
GAA P10253 1/20 0.35
MAPT P10636 1/20 0.35
PTGDR Q13258 2/20 0.35
MAP4K4 O95819 1/20 0.35
JAK2 O60674 1/20 0.35
MLNR O43193 1/20 0.35
CYP2D6 P10635 1/20 0.35
SYK P43405 1/20 0.35
PTGS1 P23219 2/20 0.34
PTGS2 P35354 2/20 0.34
EPHX2 P34913 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3528428 0.82 TSHR (0.45) ALDH1A1GPR119KDM4EGAAMAPT
SCHEMBL15449639 0.81 ALDH1A1 (0.69) ALDH1A1KCNH2CHRNA7PTGDRMLNR
SCHEMBL1853273 0.74 SYK (0.39) CHRNA7LRRK2KDM4EGAAMAPT
SCHEMBL4688848 0.73 KMT2A (0.50)
SCHEMBL14480256 0.72 ACACB (0.36) ALDH1A1NNMTKDM4EMAPTACACB
SCHEMBL1688213 0.72 KCNH2 (0.56) ALDH1A1KCNH2NNMTKDM4EPTGS1
SCHEMBL3077690 0.70 ALDH1A1 (0.67) ALDH1A1CHRNA7KDM4EPTGDRMLNR
SCHEMBL4687908 0.70 SMN1; SMN2 (0.43) ALDH1A1KDM4E
SCHEMBL13589489 0.70 CA12 (0.45) ALDH1A1KCNH2GPR119MAPTPTGS1
SCHEMBL2697225 0.69 KMT2A (0.47) ALDH1A1NNMTLRRK2KDM4EMAP4K4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1496838-A4 SUBSTITUTED AMIDES MERCK & CO INC (US) 2008-07-02 EP disclosed
EP-1496838-A2 SUBSTITUTED AMIDES Merck & Co., Inc. (US) 2005-01-19 EP disclosed
WO-2003077847-A2 SUBSTITUTED AMIDES MERCK & CO., INC. (US) 2003-09-25 WO disclosed