SCHEMBL4690503

SCHEMBL4690503

NCCN(C1CCN(CCO[PH2]=O)CC1)S(=O)(=O)c1ccc(Nc2nccc(Nc3ccc(F)c(F)c3)n2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 4/20 0.39
CDK4 P11802 1/20 0.39
CCNE1 P24864 1/20 0.39
IKBKB O14920 1/20 0.38
CHUK O15111 1/20 0.38
CA2 P00918 4/20 0.37
CA1 P00915 3/20 0.37
JAK2 O60674 2/20 0.36
JAK3 P52333 2/20 0.36
HTR1A P08908 4/20 0.36
DRD2 P14416 4/20 0.36
HTR2A P28223 4/20 0.36
HTR7 P34969 4/20 0.36
KDR P35968 2/20 0.35
EGFR P00533 1/20 0.35
INSR P06213 1/20 0.35
IGF1R P08069 1/20 0.35
MET P08581 1/20 0.35
TEK Q02763 1/20 0.35
HRH3 Q9Y5N1 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4876637 0.86 CDK2 (0.39) CDK2CDK4CCNE1IKBKBCHUK
SCHEMBL14020190 0.84 CDK2 (0.38) CDK2CDK4CCNE1IKBKBCHUK
SCHEMBL4623336 0.83 HTR1A (0.42) CDK2CDK4CCNE1CA2CA1
SCHEMBL14020182 0.82 IKBKB (0.47) CDK2CDK4CCNE1IKBKBCHUK
SCHEMBL4882378 0.82 CDK2 (0.38) CDK2CDK4CCNE1IKBKBCHUK
SCHEMBL4623334 0.82 HTR1A (0.41) CDK2CDK4CCNE1CA2CA1
SCHEMBL4623357 0.81 JAK2 (0.48) CDK2CDK4CCNE1CA2CA1
SCHEMBL14020201 0.81 CDK2 (0.38) CDK2CDK4CCNE1IKBKBCHUK
Hydrochloric Acid SCHEMBL4881375 0.80 JAK2 (0.47) CDK2CDK4CCNE1CA2CA1
SCHEMBL4621951 0.80 MEN1 (0.47) CDK2CDK4CCNE1CA2CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1904479-A2 NOVEL 2,4-DIANILINOPYRIMIDINE DERIVATIVES, THE PREPARATION THEREOF, THEIR USE AS MEDICAMENTS, PHARMACEUTICAL COMPOSITIONS AND, IN PARTICULAR, AS IKK INHIBITORS Sanofi-Aventis (FR) 2008-04-02 EP disclosed
WO-2007006926-A2 NOVEL 2,4-DIANILINOPYRIMIDINE DERIVATIVES, THE PREPARATION THEREOF, THEIR USE AS MEDICAMENTS, PHARMACEUTICAL COMPOSITIONS AND, IN PARTICULAR, AS IKK INHIBITORS SANOFI-AVENTIS (FR) 2007-01-18 WO disclosed