SCHEMBL4690664

SCHEMBL4690664

CC(=O)c1ccccc1C(=O)N1CC2CN(CCCNC(=O)c3ccc(C)c(Cl)c3)CC2C1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMYD2 Q9NRG4 2/20 0.43
SLC6A4 P31645 4/20 0.42
SLC6A2 P23975 3/20 0.42
KDM4E B2RXH2 3/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
GAA P10253 1/20 0.42
DRD2 P14416 3/20 0.42
DRD3 P35462 3/20 0.42
DRD4 P21917 2/20 0.42
ADRA1A P35348 2/20 0.42
TMEM97 Q5BJF2 1/20 0.41
SIGMAR1 Q99720 1/20 0.41
LMNA P02545 2/20 0.41
NPC1 O15118 1/20 0.41
MAPK14 Q16539 1/20 0.41
ALDH1A1 P00352 1/20 0.40
TSHR P16473 1/20 0.40
MAPK1 P28482 1/20 0.40
MAPT P10636 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4693332 0.93 SLC6A4 (0.45) SMYD2SLC6A4SLC6A2KDM4ESMN1; SMN2
SCHEMBL4693959 0.90 HCRTR1 (0.45) SMYD2SLC6A4SLC6A2KDM4ESMN1; SMN2
SCHEMBL4691761 0.90 SLC6A2 (0.44) SMYD2SLC6A4SLC6A2SMN1; SMN2DRD2
SCHEMBL4692672 0.89 SMYD2 (0.45) SMYD2SLC6A4SLC6A2SMN1; SMN2DRD2
SCHEMBL4691221 0.89 L3MBTL3 (0.45) SMYD2SMN1; SMN2GAALMNAMAPK14
SCHEMBL4691639 0.89 SMYD2 (0.48) SMYD2SLC6A4SLC6A2KDM4ESMN1; SMN2
SCHEMBL4692216 0.88 SLC6A2 (0.43) SMYD2SLC6A4SLC6A2KDM4ESMN1; SMN2
SCHEMBL3284096 0.88 SMYD2 (0.44) SMYD2SLC6A4SLC6A2KDM4ESMN1; SMN2
SCHEMBL4694269 0.87 HCRTR1 (0.48) SMYD2SLC6A4SMN1; SMN2GAADRD2
SCHEMBL4690666 0.87 NTRK1 (0.44) SLC6A4SMN1; SMN2GAADRD2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed