SCHEMBL4690858

SCHEMBL4690858

O=C(N[C@@H](CCN1CC2=CN(C(=O)c3c(F)cccc3Cl)CC2C1)c1ccccc1)c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 12/20 0.48
UTS2R Q9UKP6 5/20 0.46
ROCK2 O75116 1/20 0.41
ROCK1 Q13464 1/20 0.41
DGAT2 Q96PD7 1/20 0.38
SIGMAR1 Q99720 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4694765 0.96 CCR5 (0.44) CCR5UTS2RROCK2ROCK1DGAT2
SCHEMBL4691949 0.96 UTS2R (0.49) CCR5UTS2RROCK2ROCK1DGAT2
SCHEMBL4691249 0.95 CCR5 (0.44) CCR5UTS2RROCK2ROCK1DGAT2
SCHEMBL4690226 0.95 CCR5 (0.46) CCR5UTS2RSIGMAR1
SCHEMBL4692986 0.94 ROCK1 (0.47) CCR5UTS2RROCK2ROCK1DGAT2
SCHEMBL4696387 0.94 CCR5 (0.47) CCR5UTS2RROCK2ROCK1
SCHEMBL4690242 0.94 CCR5 (0.43) CCR5UTS2RROCK2ROCK1DGAT2
SCHEMBL4694537 0.93 CCR5 (0.44) CCR5UTS2RROCK2ROCK1DGAT2
SCHEMBL4696133 0.93 CCR5 (0.46) CCR5UTS2RDGAT2
SCHEMBL4694186 0.93 CCR5 (0.42) CCR5UTS2RROCK2ROCK1DGAT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed