SCHEMBL4692365

SCHEMBL4692365

CC(c1ccc(Cl)cc1)C(CNC(=O)C(C)(C)Oc1ccc(Cl)cc1)c1ccccn1

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.52
CNR1 P21554 13/20 0.48
CNR2 P34972 8/20 0.48
USP2 O75604 1/20 0.45
POLB P06746 1/20 0.45
MAPT P10636 1/20 0.45
HTT P42858 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
LMNA P02545 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4692132 0.95 CNR1 (0.52) ALDH1A1CNR1CNR2
SCHEMBL2653467 0.85 CNR1 (0.62) ALDH1A1CNR1CNR2USP2POLB
SCHEMBL4691613 0.85 CNR1 (0.62) ALDH1A1CNR1CNR2USP2POLB
SCHEMBL4688668 0.85 CNR1 (0.61) ALDH1A1CNR1CNR2USP2POLB
SCHEMBL4690861 0.84 CNR1 (0.63) ALDH1A1CNR1CNR2USP2POLB
SCHEMBL4688836 0.84 CNR1 (0.60) CNR1CNR2
SCHEMBL4695337 0.84 CNR1 (0.58) CNR1CNR2CYP2D6CYP2C9
SCHEMBL4688723 0.84 CNR1 (0.62) ALDH1A1CNR1CNR2
SCHEMBL4693315 0.83 CYP1A2 (0.56) ALDH1A1CNR1CNR2USP2POLB
SCHEMBL2652057 0.83 CNR1 (0.62) CNR1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1496838-A4 SUBSTITUTED AMIDES MERCK & CO INC (US) 2008-07-02 EP claimed
EP-1496838-A2 SUBSTITUTED AMIDES Merck & Co., Inc. (US) 2005-01-19 EP claimed
WO-2003077847-A2 SUBSTITUTED AMIDES MERCK & CO., INC. (US) 2003-09-25 WO claimed
EP-1496838-A4 SUBSTITUTED AMIDES MERCK & CO INC (US) 2008-07-02 EP disclosed
EP-1496838-A2 SUBSTITUTED AMIDES Merck & Co., Inc. (US) 2005-01-19 EP disclosed
WO-2003077847-A2 SUBSTITUTED AMIDES MERCK & CO., INC. (US) 2003-09-25 WO disclosed