SCHEMBL4695337

SCHEMBL4695337

CC(c1ccc(Cl)cc1)C(CNC(=O)C(C)(C)Oc1ccc(C(F)(F)F)cn1)c1ccccn1

nearest known ligand 0.58

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 18/20 0.58
CNR2 P34972 4/20 0.58
CYP2D6 P10635 1/20 0.50
CYP2C9 P11712 1/20 0.50
KCNH2 Q12809 1/20 0.50
DGAT2 Q96PD7 1/20 0.41
SCN9A Q15858 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4688817 0.90 CNR1 (0.69) CNR1CNR2CYP2D6CYP2C9KCNH2
SCHEMBL2654225 0.87 CNR1 (0.58) CNR1CNR2CYP2D6CYP2C9KCNH2
SCHEMBL4688751 0.86 CNR1 (0.60) CNR1CNR2CYP2D6CYP2C9KCNH2
SCHEMBL4692225 0.86 CNR1 (0.60) CNR1CNR2CYP2D6CYP2C9KCNH2
SCHEMBL2651795 0.84 CNR1 (0.59) CNR1CNR2CYP2D6CYP2C9KCNH2
SCHEMBL4688432 0.84 CNR1 (0.59) CNR1CNR2CYP2D6CYP2C9KCNH2
SCHEMBL1571723 0.84 CNR1 (0.55) CNR1CNR2CYP2D6CYP2C9KCNH2
SCHEMBL4692365 0.84 ALDH1A1 (0.52) CNR1CNR2CYP2D6CYP2C9
SCHEMBL4690869 0.84 CNR1 (0.71) CNR1CNR2CYP2D6CYP2C9KCNH2
SCHEMBL2653127 0.83 CNR1 (0.53) CNR1CNR2CYP2D6CYP2C9KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1496838-A4 SUBSTITUTED AMIDES MERCK & CO INC (US) 2008-07-02 EP claimed
EP-1496838-A2 SUBSTITUTED AMIDES Merck & Co., Inc. (US) 2005-01-19 EP claimed
WO-2003077847-A2 SUBSTITUTED AMIDES MERCK & CO., INC. (US) 2003-09-25 WO claimed
EP-1496838-A4 SUBSTITUTED AMIDES MERCK & CO INC (US) 2008-07-02 EP disclosed
EP-1496838-A2 SUBSTITUTED AMIDES Merck & Co., Inc. (US) 2005-01-19 EP disclosed
WO-2003077847-A2 SUBSTITUTED AMIDES MERCK & CO., INC. (US) 2003-09-25 WO disclosed