SCHEMBL4692787

SCHEMBL4692787

CCN(CC)CCC(=O)N[C@@H](CCN1CC2=CN(C(=O)c3c(F)cccc3Cl)CC2C1)c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 16/20 0.41
MAPK1 P28482 1/20 0.35
KDM4E B2RXH2 1/20 0.34
SIGMAR1 Q99720 1/20 0.34
UTS2R Q9UKP6 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4690183 0.92 CCR5 (0.43) CCR5MAPK1SIGMAR1
SCHEMBL4692079 0.90 CCR5 (0.44) CCR5MAPK1SIGMAR1UTS2R
SCHEMBL4695845 0.88 CCR5 (0.42) CCR5MAPK1SIGMAR1UTS2R
SCHEMBL4691520 0.88 CCR5 (0.42) CCR5MAPK1SIGMAR1UTS2R
SCHEMBL4691795 0.88 CCR5 (0.42) CCR5MAPK1SIGMAR1UTS2R
SCHEMBL4694571 0.87 CCR5 (0.41) CCR5SIGMAR1
SCHEMBL4693112 0.87 CCR5 (0.45) CCR5MAPK1SIGMAR1
SCHEMBL4695068 0.87 CCR5 (0.44) CCR5MAPK1SIGMAR1UTS2R
SCHEMBL4690588 0.87 CCR5 (0.48) CCR5MAPK1SIGMAR1
SCHEMBL4692327 0.86 CCR5 (0.49) CCR5SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed